SCHEMBL5099349

SCHEMBL5099349

COCCOCC(NC(C)=O)c1cc(CCCOc2c(C)cc(-c3ccccc3)cc2C)on1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 4/20 0.36
ITGB1 P05556 3/20 0.35
ITGA4 P13612 3/20 0.35
NR1I2 O75469 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
TP53 P04637 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
LIPC P11150 1/20 0.33
LIPG Q9Y5X9 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
CA12 O43570 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5099362 0.85 NR1I2 (0.39) NR1I2CYP3A4CYP2D6L3MBTL1NPC1
SCHEMBL5098199 0.84 NR1I2 (0.39) NR1I2CYP3A4CYP2D6L3MBTL1NPC1
SCHEMBL5092827 0.71 NR1I2 (0.44) NR1I2CYP3A4CYP2D6L3MBTL1NPC1
SCHEMBL5089005 0.70 NR1I2 (0.45) NR1I2CYP3A4CYP2D6L3MBTL1NPC1
SCHEMBL5088999 0.70 NR1I2 (0.42) NR1I2CYP3A4CYP2D6NPC1RAB9A
SCHEMBL7492829 0.69 NR1I2 (0.41) NR1I2CYP3A4CYP2D6L3MBTL1NPC1
SCHEMBL5098193 0.69 RAB9A (0.40) NR1I2CYP3A4CYP2D6L3MBTL1NPC1
SCHEMBL5088906 0.68 NR1I2 (0.45) NR1I2CYP3A4CYP2D6L3MBTL1NPC1
SCHEMBL7496717 0.68 HDAC6 (0.37) NR1I2CYP3A4CYP2D6HDAC1HDAC6
SCHEMBL5089011 0.68 NR1I2 (0.65) NR1I2CYP3A4CYP2D6HDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7371755-B1 Antiviral agents BIOTA SCIENTIFIC MANAGEMENT PTY LTD. (AU) 2008-05-13 US disclosed
EP-1214317-A1 ANTIVIRAL AGENTS BIOTA SCIENTIFIC MANAGEMENT PTY. LTD. (AU) 2002-06-19 EP disclosed
WO-2001019822-A1 ANTIVIRAL AGENTS BIOTA SCIENTIFIC MANAGEMENT PTY LTD (AU) 2001-03-22 WO disclosed