SCHEMBL5111718

SCHEMBL5111718

Cc1c(Cl)ccc(S(=O)(=O)N(CCCCC(=O)N(C)Cc2ccc(C3=NCCN3C(=O)O)cc2)CCC(N)=O)c1Cl

nearest known ligand 0.54

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BDKRB1 P46663 11/20 0.54
LMNA P02545 1/20 0.40
DGAT1 O75907 1/20 0.31
HTT P42858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5125768 0.94 BDKRB1 (0.54) BDKRB1LMNADGAT1
SCHEMBL5118277 0.90 BDKRB1 (0.66) BDKRB1LMNA
SCHEMBL5118841 0.88 BDKRB1 (0.69) BDKRB1LMNA
SCHEMBL5111740 0.86 BDKRB1 (0.67) BDKRB1LMNA
SCHEMBL5950333 0.85 LMNA (0.39) BDKRB1LMNA
SCHEMBL5118568 0.84 BDKRB1 (0.57) BDKRB1LMNADGAT1
SCHEMBL4030306 0.83 BDKRB1 (0.78) BDKRB1
SCHEMBL6760042 0.83 BDKRB1 (0.58) BDKRB1LMNAHTT
SCHEMBL5118845 0.81 BDKRB1 (0.50) BDKRB1LMNADGAT1
SCHEMBL5119725 0.80 BDKRB1 (0.52) BDKRB1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7361687-B2 Arylsulphonamide derivatives and methods of preparing LABORATOIRES FOURNIER SA (FR) 2008-04-22 US disclosed
US-20060084699-A1 Novel arylsulphonamide derivatives and use thereof as therapeutic agents LABORATOIRES FOURNIER SA (FR) 2006-04-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060084699-A1 Novel arylsulphonamide derivatives and use thereof as therapeutic agents UGT1A1, UGT2B7, UGT1A6 BDKRB1 1217/4885LMNA 4632/4885DGAT1 2239/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.