SCHEMBL5113516

SCHEMBL5113516

CC(C)(C)OC(=O)Nc1cc(C(=O)c2cc(CC(=O)O)c(-c3ccccc3)s2)ccc1I

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
MAPT P10636 2/20 0.44
ALDH1A1 P00352 1/20 0.44
HTT P42858 1/20 0.44
HDAC1 Q13547 1/20 0.40
RXFP1 Q9HBX9 2/20 0.38
TP53 P04637 2/20 0.38
SUCNR1 Q9BXA5 2/20 0.37
LCK P06239 2/20 0.37
NR1H4 Q96RI1 1/20 0.37
CNR2 P34972 1/20 0.36
BRD9 Q9H8M2 1/20 0.36
GLS O94925 1/20 0.33
PPARG P37231 3/20 0.33
PPARA Q07869 3/20 0.33
PPARD Q03181 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
PTGS2 P35354 1/20 0.32
AKT1 P31749 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16893446 0.73 MAPT (0.57) MEN1KMT2AMAPTALDH1A1HTT
SCHEMBL15545929 0.72 MEN1 (0.63) MEN1KMT2AMAPTALDH1A1HTT
SCHEMBL3052808 0.72 BRD4 (0.39) MEN1KMT2AMAPTALDH1A1HTT
SCHEMBL3056704 0.71 BRD4 (0.38) SUCNR1CNR2
SCHEMBL3058707 0.71 MAPT (0.40) MEN1KMT2AMAPTALDH1A1HTT
SCHEMBL3058715 0.71 KMT2A (0.55) MEN1KMT2AMAPTALDH1A1HTT
SCHEMBL16904651 0.71 MAPT (0.68) MEN1KMT2AMAPTALDH1A1HTT
SCHEMBL16893399 0.71 MEN1 (0.55) MEN1KMT2AMAPTALDH1A1HTT
SCHEMBL3042819 0.69 KMT2A (0.44) MEN1KMT2AMAPTALDH1A1HTT
SCHEMBL29281561 0.69 KDM4E (0.49) KMT2AMAPTALDH1A1HDAC1LCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008051197-A2 SMALL-MOLECULE BOTULINUM TOXIN INHIBITORS MAYO FOUNDATION FOR MEDICAL EDUCATION AND RESEARCH (US) 2008-05-02 WO disclosed