SCHEMBL5115902

SCHEMBL5115902

CNC(=O)c1cc(Oc2cccc(CCNC(=O)c3cccc(OC)c3C)c2)ccn1

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 1/20 0.48
RAF1 P04049 3/20 0.47
BRAF P15056 2/20 0.47
GPR52 Q9Y2T5 2/20 0.47
TP53 P04637 1/20 0.45
DDR2 Q16832 1/20 0.44
KDR P35968 4/20 0.44
RET P07949 1/20 0.42
TAAR1 Q96RJ0 1/20 0.42
THRA P10827 1/20 0.41
THRB P10828 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14266579 0.93 CSF1R (0.49) CSF1RRAF1BRAFTP53KDR
SCHEMBL3991259 0.91 BRAF (0.48) CSF1RRAF1BRAFTP53DDR2
SCHEMBL14266603 0.89 CSF1R (0.49) CSF1RRAF1BRAFDDR2KDR
SCHEMBL5123391 0.88 RAF1 (0.53) CSF1RRAF1BRAFDDR2KDR
SCHEMBL14266573 0.87 CSF1R (0.54) CSF1RRAF1BRAFTP53KDR
SCHEMBL3987237 0.87 BRAF (0.50) RAF1BRAFKDRRET
SCHEMBL3989617 0.86 KDR (0.47) CSF1RRAF1BRAFDDR2KDR
SCHEMBL5123752 0.86 KMT2A (0.51) CSF1RRAF1BRAFKDR
SCHEMBL14266542 0.86 DDR2 (0.51) CSF1RRAF1BRAFTP53DDR2
SCHEMBL5128896 0.86 DNMT3A (0.54) CSF1RRAF1BRAFDDR2KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080064729-A1 Phenethylamide derivatives with kinase inhibitory activity MILLENNIUM PHARMACEUTICALS, INC. (US) 2008-03-13 US disclosed
US-20080064729-A1 Phenethylamide derivatives with kinase inhibitory activity MILLENNIUM PHARMACEUTICALS, INC. (US) 2008-03-13 US disclosed
US-20080064729-A1 Phenethylamide derivatives with kinase inhibitory activity MILLENNIUM PHARMACEUTICALS, INC. (US) 2008-03-13 US disclosed
WO-2008030448-A1 PHENETHYLAMIDE DERIVATIVES WITH KINASE INHIBITORY ACTIVITY MILLENNIUM PHARMACEUTICALS, INC. (US) 2008-03-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080064729-A1 Phenethylamide derivatives with kinase inhibitory activity MAP4K5, MAP3K5, MAP4K2 CSF1R 2904/4885RAF1 251/4885BRAF 242/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.