SCHEMBL5119787

SCHEMBL5119787

O=C1NC(=S)S/C1=C/c1ccc(-c2cc(Cl)cc(Cl)c2)o1

nearest known ligand 0.65

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
IGF1R P08069 5/20 0.65
INSR P06213 4/20 0.65
DNM1 Q05193 1/20 0.62
PIK3CG P48736 5/20 0.61
GSK3A P49840 3/20 0.61
GSK3B P49841 3/20 0.61
HSPD1 P10809 1/20 0.58
HSPE1 P61604 1/20 0.58
PTP4A3 O75365 1/20 0.55
PIM1 P11309 2/20 0.54
MYC P01106 1/20 0.53
NAT1 P18440 1/20 0.53
MAX P61244 1/20 0.53
PIK3CA P42336 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5119790 1.00 IGF1R (0.65) IGF1RINSRDNM1PIK3CGGSK3A
SCHEMBL14411129 1.00 IGF1R (0.65) IGF1RINSRDNM1PIK3CGGSK3A
SCHEMBL623749 0.89 GSK3A (0.77) IGF1RINSRPIK3CGGSK3AGSK3B
SCHEMBL623748 0.89 GSK3A (0.77) IGF1RINSRPIK3CGGSK3AGSK3B
SCHEMBL623750 0.89 GSK3A (0.77) IGF1RINSRPIK3CGGSK3AGSK3B
SCHEMBL14277838 0.88 IGF1R (0.73) IGF1RINSRPIK3CGGSK3AGSK3B
SCHEMBL6089724 0.88 IGF1R (0.72) IGF1RINSRPIK3CGGSK3AGSK3B
SCHEMBL3904134 0.88 IGF1R (0.72) IGF1RINSRPIK3CGGSK3AGSK3B
SCHEMBL3904132 0.88 IGF1R (0.72) IGF1RINSRPIK3CGGSK3AGSK3B
SCHEMBL5124788 0.85 IGF1R (0.80) IGF1RINSRPIK3CGGSK3AGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080051445-A1 2-Thioxothiazolidin-4-one compounds and compositions as antimicrobial and antimalarial agents targeting enoyl-ACP reductase of type II fatty acid synthesis pathway and other cell growth pathways NATIONAL INSTITUTE OF IMMUNOLOGY. 2008-02-28 US disclosed
EP-1834642-A2 2-thioxothiazolidin-4-one compounds and compositions as antimicrobial and antimalarial agents targeting enoyl-ACP reductase of type II fatty acid synthesis pathway and other cell growth pathways National Institute of Immunology (IN) 2007-09-19 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080051445-A1 2-Thioxothiazolidin-4-one compounds and compositions as antimicrobial and antimalarial agents targeting enoyl-ACP reductase of type II fatty acid synthesis pathway and other cell growth pathways FASN, FADS2, TECR IGF1R 3557/4885INSR 2530/4885DNM1 3032/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.