SCHEMBL5128332

SCHEMBL5128332

COCC(=O)N[C@H](C)C(N)=O

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.44
SMN1; SMN2 Q16637 2/20 0.40
HPGD P15428 2/20 0.40
RECQL P46063 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
NPSR1 Q6W5P4 1/20 0.36
ALDH1A1 P00352 2/20 0.36
KDM4E B2RXH2 1/20 0.36
ACACB O00763 2/20 0.35
ACACA Q13085 1/20 0.35
CA14 Q9ULX7 1/20 0.33
LMNA P02545 1/20 0.33
PSMB5 P28074 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9954665 1.00 TSHR (0.44) TSHRSMN1; SMN2HPGDRECQLMEN1
SCHEMBL3673890 0.85 TSHR (0.50) TSHRSMN1; SMN2HPGDRECQLMEN1
SCHEMBL3673892 0.85 TSHR (0.50) TSHRSMN1; SMN2HPGDRECQLMEN1
SCHEMBL28127289 0.85 TSHR (0.50) TSHRSMN1; SMN2HPGDRECQLMEN1
SCHEMBL19036963 0.83 KDM4E (0.35) TSHRSMN1; SMN2RECQLMEN1KMT2A
SCHEMBL31308086 0.83 TSHR (0.36) TSHRSMN1; SMN2RECQLMEN1KMT2A
SCHEMBL3397754 0.81 SMN1; SMN2 (0.51) TSHRSMN1; SMN2HPGDNPSR1ALDH1A1
SCHEMBL2294082 0.81 SMN1; SMN2 (0.51) TSHRSMN1; SMN2HPGDNPSR1ALDH1A1
SCHEMBL25646522 0.81 TSHR (0.46) TSHRSMN1; SMN2HPGDRECQLMEN1
SCHEMBL2294079 0.81 SMN1; SMN2 (0.51) TSHRSMN1; SMN2HPGDNPSR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080161325-A1 e.g. N1-[3-amino-4-(3,5-difluorophenyl)-2-hydroxybutyl]-3-(butylsulfonyl)-N1-(3-ethylbenzyl)-D-alaninamide dihydrochloride; inhibitors of amyloid beta-secretase enzyme; neurodegenerative diseases: Alzheimer's, Parkinson's diseases, Down's syndrome ELAN PHARMACEUTICALS, INC. 2008-07-03 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080161325-A1 e.g. N1-[3-amino-4-(3,5-difluorophenyl)-2-hydroxybutyl]-3-(butylsulfonyl)-N1-(3-ethylbenzyl)-D-alaninamide dihydrochloride; inhibitors of amyloid beta-secretase enzyme; neurodegenerative diseases: Alzheimer's, Parkinson's diseases, Down's syndrome BACE1, APP, BACE2 TSHR 4721/4885SMN1; SMN2 154/4885HPGD 1263/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.