SCHEMBL5131133

SCHEMBL5131133

CCCN(CCC)S(=O)(=O)CCC(=O)O[C@H](CNCCC(C)C)[C@@H](N)Cc1cc(F)cc(OCc2ccccc2)c1

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 6/20 0.39
CTSD P07339 4/20 0.39
REN P00797 1/20 0.34
MMP2 P08253 2/20 0.33
MMP13 P45452 2/20 0.33
ADAMTS4 O75173 1/20 0.33
MMP14 P50281 1/20 0.33
ADAMTS5 Q9UNA0 1/20 0.33
LTA4H P09960 1/20 0.33
LAP3 P28838 3/20 0.32
ANPEP P15144 1/20 0.32
RNPEP Q9H4A4 1/20 0.32
DNPEP Q9ULA0 1/20 0.32
ABCB1 P08183 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5131136 1.00 BACE1 (0.39) BACE1CTSDRENMMP2MMP13
SCHEMBL5124815 0.88 BACE1 (0.55) BACE1CTSD
SCHEMBL5124820 0.88 BACE1 (0.55) BACE1CTSD
Hydrochloric Acid SCHEMBL5131063 0.87 BACE1 (0.54) BACE1CTSD
SCHEMBL5117493 0.85 CTSD (0.32) BACE1CTSD
SCHEMBL5117495 0.85 CTSD (0.32) BACE1CTSD
SCHEMBL5130561 0.83 CTSD (0.41) BACE1CTSD
SCHEMBL5130558 0.83 CTSD (0.41) BACE1CTSD
SCHEMBL3346884 0.82 BACE1 (0.60) BACE1CTSD
SCHEMBL3346879 0.82 BACE1 (0.60) BACE1CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080161325-A1 e.g. N1-[3-amino-4-(3,5-difluorophenyl)-2-hydroxybutyl]-3-(butylsulfonyl)-N1-(3-ethylbenzyl)-D-alaninamide dihydrochloride; inhibitors of amyloid beta-secretase enzyme; neurodegenerative diseases: Alzheimer's, Parkinson's diseases, Down's syndrome ELAN PHARMACEUTICALS, INC. 2008-07-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080161325-A1 e.g. N1-[3-amino-4-(3,5-difluorophenyl)-2-hydroxybutyl]-3-(butylsulfonyl)-N1-(3-ethylbenzyl)-D-alaninamide dihydrochloride; inhibitors of amyloid beta-secretase enzyme; neurodegenerative diseases: Alzheimer's, Parkinson's diseases, Down's syndrome BACE1, APP, BACE2 BACE1 1/4885CTSD 100/4885REN 1107/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.