SCHEMBL5133499

SCHEMBL5133499

O=C(C=Cc1ccc2nc[nH]c2c1)NO

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 12/20 1.00
HDAC6 Q9UBN7 2/20 0.65
GPR183 P32249 1/20 0.51
HDAC8 Q9BY41 3/20 0.50
ESR1 P03372 1/20 0.48
HDAC2 Q92769 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3366897 0.89 HDAC1 (0.80) HDAC1HDAC6HDAC8HDAC2
SCHEMBL3366899 0.89 HDAC1 (0.80) HDAC1HDAC6HDAC8HDAC2
SCHEMBL4574406 0.82 HDAC1 (0.70) HDAC1HDAC6GPR183ESR1
SCHEMBL4572978 0.82 HDAC1 (0.70) HDAC1HDAC6GPR183ESR1
SCHEMBL18469368 0.78 HDAC1 (0.63) HDAC1
SCHEMBL15552440 0.78 HDAC1 (0.63) HDAC1
SCHEMBL10817405 0.75 IP6K1 (0.63) HDAC1HDAC6ESR1
SCHEMBL30050466 0.75 IP6K1 (0.63) HDAC1HDAC6ESR1
SCHEMBL14972936 0.75 IP6K1 (0.63) HDAC1HDAC6ESR1
SCHEMBL16215254 0.75 HDAC1 (0.58) HDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1673349-A4 BENZIMIDAZOLE DERIVATES: PREPARATION AND PHARMACEUTICAL APPLICATIONS S BIO PTE LTD (SG) 2008-01-23 EP disclosed
EP-1673349-A1 BENZIMIDAZOLE DERIVATES: PREPARATION AND PHARMACEUTICAL APPLICATIONS S*Bio Pte Ltd (SG) 2006-06-28 EP disclosed
WO-2005028447-A1 BENZIMIDAZOLE DERIVATES: PREPARATION AND PHARMACEUTICAL APPLICATIONS S*BIO PTE LTD (SG) 2005-03-31 WO disclosed