SCHEMBL5133685

SCHEMBL5133685

OCCCn1c(Sc2ccc3c(c2)OCCO3)nc2c([AsH2])ncnc21

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 15/20 0.42
HSP90AB1 P08238 14/20 0.42
HSP90B1 P14625 7/20 0.41
ERBB2 P04626 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
HDAC3 O15379 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC7 Q8WUI4 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC10 Q969S8 1/20 0.38
HDAC11 Q96DB2 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
HDAC9 Q9UKV0 1/20 0.38
HDAC5 Q9UQL6 1/20 0.38
TRAP1 Q12931 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5142341 0.94 HSP90AA1 (0.47) HSP90AA1HSP90AB1HSP90B1ERBB2HDAC3
SCHEMBL5132561 0.89 HSP90AA1 (0.54) HSP90AA1HSP90AB1HSP90B1ERBB2TRAP1
SCHEMBL5131899 0.83 HSP90AA1 (0.59) HSP90AA1HSP90AB1HSP90B1ERBB2HDAC3
SCHEMBL5035593 0.76 HSP90AA1 (0.56) HSP90AA1HSP90AB1HSP90B1HDAC3HDAC4
SCHEMBL3465421 0.73 HSP90AA1 (0.66) HSP90AA1HSP90AB1HSP90B1ERBB2HDAC3
SCHEMBL3124067 0.71 HSP90AA1 (0.54) HSP90AA1HSP90AB1HSP90B1ERBB2HDAC3
SCHEMBL5130186 0.71 HSP90AB1 (0.56) HSP90AA1HSP90AB1HSP90B1ERBB2HDAC3
SCHEMBL3124508 0.71 HSP90AB1 (0.57) HSP90AA1HSP90AB1HSP90B1ERBB2HDAC3
SCHEMBL13731589 0.70 HSP90AA1 (0.65) HSP90AA1HSP90AB1
SCHEMBL15980449 0.69 HSP90AA1 (0.74) HSP90AA1HSP90AB1HSP90B1ERBB2HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1962863-A2 ORALLY ACTIVE PURINE-BASED INHIBITORS OF HEAT SHOCK PROTEIN 90 Conforma Therapeutics Corporation (US) 2008-09-03 EP disclosed
WO-2007075572-A2 ORALLY ACTIVE PURINE-BASED INHIBITORS OF HEAT SHOCK PROTEIN 90 CONFORMA THERAPEUTICS CORPORATION (US) 2007-07-05 WO disclosed