SCHEMBL5133764

SCHEMBL5133764

CC1CN(C(C)c2cc(F)c(F)c(F)c2)CCN1

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.35
XIAP P98170 4/20 0.33
BIRC2 Q13490 3/20 0.33
CHRM4 P08173 1/20 0.31
KDM4E B2RXH2 2/20 0.31
ALDH1A1 P00352 2/20 0.31
HPGD P15428 2/20 0.31
HSD17B10 Q99714 2/20 0.31
PMP22 Q01453 1/20 0.31
CACNA2D1 P54289 3/20 0.30
OPRM1 P35372 1/20 0.30
DGKA P23743 1/20 0.30
DGKZ Q13574 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4094000 1.00 HRH3 (0.35) HRH3XIAPBIRC2CHRM4KDM4E
SCHEMBL4102926 1.00 HRH3 (0.35) HRH3XIAPBIRC2CHRM4KDM4E
SCHEMBL4982738 0.86 HRH3 (0.38) HRH3XIAPBIRC2CACNA2D1OPRM1
SCHEMBL4107027 0.86 HRH3 (0.38) HRH3XIAPBIRC2CACNA2D1OPRM1
SCHEMBL4100180 0.86 HRH3 (0.38) HRH3XIAPBIRC2CACNA2D1OPRM1
SCHEMBL4093102 0.85 HRH3 (0.39) HRH3XIAPBIRC2CACNA2D1OPRM1
SCHEMBL4094531 0.85 HRH3 (0.39) HRH3XIAPBIRC2CACNA2D1OPRM1
SCHEMBL4099431 0.81 HRH3 (0.34) HRH3XIAPBIRC2
SCHEMBL5133237 0.81 HRH3 (0.34) HRH3XIAPBIRC2
SCHEMBL4097155 0.81 HRH3 (0.34) HRH3XIAPBIRC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008134036-A1 ALPHA-SUBSTITUTED ARYLMETHYL PIPERAZINE PYRAZOLO[1,5-α]PYRIMIDINE AMIDE DERIVATIVES PANACOS PHARMACEUTICALS, INC. (US) 2008-11-06 WO disclosed