SCHEMBL5133879

SCHEMBL5133879

CC(C)(C)OC(=O)n1c(-c2cc(OCCCN3CCC[C@H]3CO)c(Cl)c3c[nH]cc23)cc2cc(CN3CCCCC3)ccc21

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 11/20 0.33
ACHE P22303 2/20 0.33
NR1H2 P55055 2/20 0.33
ATR Q13535 2/20 0.32
ATRIP Q8WXE1 2/20 0.32
INSR P06213 1/20 0.32
ITK Q08881 1/20 0.32
F2 P00734 1/20 0.32
AURKA O14965 1/20 0.32
RPS6KB1 P23443 1/20 0.32
AURKB Q96GD4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3048852 0.88 HRH3 (0.32) HRH3ACHENR1H2
SCHEMBL3048856 0.88 HRH3 (0.32) HRH3ACHENR1H2
SCHEMBL27720805 0.87 HRH3 (0.31) HRH3ACHENR1H2
SCHEMBL5140104 0.85 NR1H2 (0.34) HRH3NR1H2ATRATRIP
SCHEMBL3042343 0.77 HRH3 (0.42) HRH3ACHE
SCHEMBL27700295 0.77 HRH3 (0.42) HRH3ACHE
SCHEMBL3044021 0.76 HRH3 (0.41) HRH3ACHEAURKA
SCHEMBL28772335 0.75 HRH3 (0.41) HRH3ACHE
SCHEMBL28943660 0.75 HRH3 (0.38) HRH3ACHEATRATRIP
SCHEMBL3159224 0.74 HRH3 (0.39) HRH3ATRATRIPAURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1880993-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND KYOWA HAKKO KOGYO CO., LTD. (JP) 2008-01-23 EP disclosed