SCHEMBL5140104

SCHEMBL5140104

CC(C)(CO)NCCCOc1cc(-c2cc3cc(CN4CCCCC4)ccc3n2C(=O)OC(C)(C)C)c2c[nH]cc2c1Cl

nearest known ligand 0.36

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 6/20 0.34
ATR Q13535 2/20 0.33
ATRIP Q8WXE1 2/20 0.33
TBK1 Q9UHD2 1/20 0.32
HRH3 Q9Y5N1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3042563 0.86 TBK1 (0.32) NR1H2ATRATRIPTBK1
SCHEMBL5133879 0.85 HRH3 (0.33) NR1H2ATRATRIPHRH3
SCHEMBL3052537 0.77 PARP1 (0.35) NR1H2TBK1HRH3
SCHEMBL3043946 0.77 NR1H2 (0.34) NR1H2TBK1HRH3
SCHEMBL3046394 0.76 NR1H2 (0.33) NR1H2ATRATRIPTBK1HRH3
SCHEMBL5133804 0.76 DRD2 (0.36) NR1H2ATRATRIP
SCHEMBL3048541 0.76 NR1H2 (0.35) NR1H2ATRATRIPTBK1
SCHEMBL27700218 0.76 NR1H2 (0.33) NR1H2HRH3
SCHEMBL3043777 0.75 HRH3 (0.33) HRH3
SCHEMBL3042568 0.75 TBK1 (0.31) NR1H2ATRATRIPTBK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1880993-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND KYOWA HAKKO KOGYO CO., LTD. (JP) 2008-01-23 EP disclosed