SCHEMBL5134593

SCHEMBL5134593

NCc1ccc(C(=O)Nc2nn(-c3ccccc3)cc2N)cc1.Nc1cn(-c2ccccc2)nc1NC(=O)c1ccc(CNC(=O)O)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
TSHR P16473 1/20 0.49
CYP2C19 P33261 1/20 0.49
HDAC1 Q13547 11/20 0.48
ADORA3 P0DMS8 3/20 0.45
KLKB1 P03952 1/20 0.45
HDAC2 Q92769 3/20 0.44
HDAC3 O15379 2/20 0.44
HDAC4 P56524 2/20 0.44
HDAC7 Q8WUI4 2/20 0.44
HDAC8 Q9BY41 2/20 0.44
HDAC6 Q9UBN7 2/20 0.44
HDAC9 Q9UKV0 2/20 0.44
HDAC5 Q9UQL6 2/20 0.44
KMT2A Q03164 2/20 0.44
MIF P14174 1/20 0.44
MEN1 O00255 1/20 0.44
HDAC10 Q969S8 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4453120 0.96 HDAC1 (0.52) HDAC1ADORA3HDAC2HDAC3HDAC4
SCHEMBL2441079 0.92 HDAC1 (0.47) HDAC1ADORA3HDAC2HDAC3
SCHEMBL14312496 0.88 ADORA3 (0.53) CYP1A2CYP2D6CYP2C9TSHRCYP2C19
SCHEMBL14312607 0.88 HDAC1 (0.53) HDAC1ADORA3HDAC2HDAC3HDAC4
SCHEMBL14312488 0.87 ADORA3 (0.49) HDAC1ADORA3KMT2AMIFMEN1
SCHEMBL14312442 0.87 HDAC1 (0.54) HDAC1ADORA3HDAC2HDAC3HDAC4
SCHEMBL14312583 0.86 HDAC1 (0.50) HDAC1HDAC2HDAC3MIF
SCHEMBL14312744 0.85 HDAC1 (0.55) TSHRHDAC1ADORA3HDAC2HDAC3
SCHEMBL14312420 0.85 HDAC1 (0.46) HDAC1ADORA3HDAC2HDAC3HDAC4
SCHEMBL14312860 0.85 HDAC1 (0.54) HDAC1ADORA3HDAC2HDAC3HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1945617-A2 HISTONE DEACETYLASE INHIBITORS WITH ARYL-PYRAZOLYL MOTIFS Merck & Co., Inc. (US) 2008-07-23 EP disclosed
WO-2007055941-A2 HISTONE DEACETYLASE INHIBITORS WITH ARYL-PYRAZOLYL MOTIFS MERCK & CO., INC. (US) 2007-05-18 WO disclosed