SCHEMBL5134787

SCHEMBL5134787

CCCCn1c(CN(CCc2ccccc2)Cc2ccc(OC)cc2)cnc1-c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
BCHE P06276 4/20 0.42
HSD11B1 P28845 2/20 0.41
SMPD1 P17405 2/20 0.40
TSHR P16473 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
KCNH2 Q12809 1/20 0.37
SIGMAR1 Q99720 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5138093 0.93 TSHR (0.43) HSD11B1SMPD1TSHRL3MBTL1
SCHEMBL5135920 0.92 BCHE (0.44) BCHEHSD11B1TSHR
SCHEMBL5075074 0.92 TSHR (0.46) BCHEHSD11B1TSHR
SCHEMBL5072355 0.91 HSD11B1 (0.45) BCHEHSD11B1TSHRL3MBTL1
SCHEMBL5135239 0.91 BCHE (0.47) BCHESIGMAR1
SCHEMBL5135667 0.90 HSD11B1 (0.44) BCHEHSD11B1TSHRL3MBTL1
SCHEMBL5134920 0.90 HSD11B1 (0.44) BCHEHSD11B1TSHRKCNH2
SCHEMBL5073933 0.88 HSD11B1 (0.43) BCHEHSD11B1TSHRL3MBTL1
SCHEMBL5137544 0.87 HSP90AA1 (0.39) BCHETSHRL3MBTL1
SCHEMBL5072318 0.87 TSHR (0.40) HSD11B1SMPD1TSHRL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1490044-A4 COMBINATION THERAPY FOR THE TREATMENT OF CONDITIONS WITH PATHOGENIC INFLAMMATORY COMPONENTS NEUROGEN CORP (US) 2008-04-16 EP disclosed
EP-1490044-A1 COMBINATION THERAPY FOR THE TREATMENT OF CONDITIONS WITH PATHOGENIC INFLAMMATORY COMPONENTS NEUROGEN CORPORATION (US) 2004-12-29 EP disclosed
WO-2003084524-A1 COMBINATION THERAPY FOR THE TREATMENT OF CONDITIONS WITH PATHOGENIC INFLAMMATORY COMPONENTS NEUROGEN CORPORATION (US) 2003-10-16 WO disclosed