SCHEMBL5135658

SCHEMBL5135658

CCCCn1c(CN(CCc2cccc(OC)c2)Cc2ccc3c(c2)OCO3)cnc1-c1ccc(F)cc1

nearest known ligand 0.57

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 6/20 0.52
HTR2C P28335 6/20 0.52
HTR2B P41595 6/20 0.52
CTSL P07711 1/20 0.47
POLB P06746 2/20 0.45
GAA P10253 1/20 0.45
MAPT P10636 1/20 0.45
TP53 P04637 4/20 0.43
C5AR1 P21730 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5135288 0.94 HTR2A (0.51) HTR2AHTR2CHTR2BCTSLPOLB
SCHEMBL5137845 0.93 HTR2A (0.54) HTR2AHTR2CHTR2BCTSLPOLB
SCHEMBL5136838 0.93 HTR2A (0.46) HTR2AHTR2CHTR2BCTSLPOLB
SCHEMBL5136744 0.92 C5AR1 (0.47) HTR2AHTR2CHTR2BCTSLPOLB
SCHEMBL5136702 0.90 C5AR1 (0.51) HTR2AHTR2CHTR2BCTSLPOLB
SCHEMBL5136215 0.90 HTR2A (0.57) HTR2AHTR2CHTR2BTP53SMN1; SMN2
SCHEMBL5136286 0.89 HTR2A (0.48) HTR2AHTR2CHTR2BPOLBGAA
SCHEMBL5135206 0.89 TP53 (0.45) HTR2AHTR2CHTR2BPOLBGAA
SCHEMBL5136159 0.89 C5AR1 (0.48) HTR2AHTR2CHTR2BCTSLPOLB
SCHEMBL5136612 0.89 C5AR1 (0.45) HTR2AHTR2CHTR2BCTSLPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1490044-A4 COMBINATION THERAPY FOR THE TREATMENT OF CONDITIONS WITH PATHOGENIC INFLAMMATORY COMPONENTS NEUROGEN CORP (US) 2008-04-16 EP disclosed
EP-1490044-A1 COMBINATION THERAPY FOR THE TREATMENT OF CONDITIONS WITH PATHOGENIC INFLAMMATORY COMPONENTS NEUROGEN CORPORATION (US) 2004-12-29 EP disclosed
WO-2003084524-A1 COMBINATION THERAPY FOR THE TREATMENT OF CONDITIONS WITH PATHOGENIC INFLAMMATORY COMPONENTS NEUROGEN CORPORATION (US) 2003-10-16 WO disclosed