SCHEMBL5135288

SCHEMBL5135288

CCCCn1c(CN(CCc2cccc(OC)c2)Cc2ccc3c(c2)OCO3)cnc1-c1cccc(F)c1

nearest known ligand 0.57

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 6/20 0.51
HTR2C P28335 6/20 0.51
HTR2B P41595 6/20 0.51
CTSL P07711 1/20 0.46
POLB P06746 1/20 0.45
GAA P10253 1/20 0.45
MAPT P10636 1/20 0.45
C5AR1 P21730 1/20 0.42
TP53 P04637 3/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
F2R P25116 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5136312 0.94 HTR2A (0.44) HTR2AHTR2CHTR2BCTSLPOLB
SCHEMBL5135658 0.94 HTR2A (0.52) HTR2AHTR2CHTR2BCTSLPOLB
SCHEMBL5137845 0.93 HTR2A (0.54) HTR2AHTR2CHTR2BCTSLPOLB
SCHEMBL5134864 0.91 HTR2A (0.57) HTR2AHTR2CHTR2BTP53SMN1; SMN2
SCHEMBL5137540 0.90 HTR2A (0.53) HTR2AHTR2CHTR2BPOLBTP53
SCHEMBL5137390 0.88 C5AR1 (0.44) HTR2AHTR2CHTR2BPOLBC5AR1
SCHEMBL4768999 0.88 C5AR1 (0.51) HTR2AHTR2CHTR2BCTSLPOLB
SCHEMBL5136966 0.88 HTR2A (0.43) HTR2AHTR2CHTR2BCTSLPOLB
SCHEMBL5136963 0.87 C5AR1 (0.47) HTR2AHTR2CHTR2BPOLBC5AR1
SCHEMBL5138029 0.87 C5AR1 (0.53) HTR2AHTR2CHTR2BCTSLGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1490044-A4 COMBINATION THERAPY FOR THE TREATMENT OF CONDITIONS WITH PATHOGENIC INFLAMMATORY COMPONENTS NEUROGEN CORP (US) 2008-04-16 EP disclosed
EP-1490044-A1 COMBINATION THERAPY FOR THE TREATMENT OF CONDITIONS WITH PATHOGENIC INFLAMMATORY COMPONENTS NEUROGEN CORPORATION (US) 2004-12-29 EP disclosed
WO-2003084524-A1 COMBINATION THERAPY FOR THE TREATMENT OF CONDITIONS WITH PATHOGENIC INFLAMMATORY COMPONENTS NEUROGEN CORPORATION (US) 2003-10-16 WO disclosed