SCHEMBL5136522

SCHEMBL5136522

O=C1OC2(CCNCC2)c2cc(CF)ccc21

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.42
NPY5R Q15761 8/20 0.38
CTSC P53634 2/20 0.37
AVPR1A P37288 3/20 0.33
DRD2 P14416 1/20 0.33
CCNC P24863 1/20 0.32
CDK8 P49336 1/20 0.32
HASPIN Q8TF76 1/20 0.32
CDK19 Q9BWU1 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6820160 0.85 SIGMAR1 (0.41) SIGMAR1NPY5RCTSCAVPR1ADRD2
SCHEMBL22057308 0.81 NPY5R (0.45) SIGMAR1NPY5RCTSCAVPR1A
Hydrochloric Acid SCHEMBL6820680 0.80 NPY5R (0.44) SIGMAR1NPY5RCTSCAVPR1ADRD2
SCHEMBL3839131 0.78 AVPR1A (0.50) SIGMAR1NPY5RAVPR1A
SCHEMBL18373156 0.78 NPY5R (0.45) SIGMAR1NPY5RCTSCAVPR1ADRD2
Hydrochloric Acid SCHEMBL6819610 0.77 AVPR1A (0.49) SIGMAR1CTSCAVPR1ADRD2CCNC
SCHEMBL29674557 0.76 SIGMAR1 (0.54) SIGMAR1NPY5RAVPR1A
SCHEMBL171980 0.76 SIGMAR1 (0.54) SIGMAR1NPY5RAVPR1A
SCHEMBL736508 0.75 AVPR1A (0.53) NPY5RAVPR1A
SCHEMBL30476248 0.75 SIGMAR1 (0.36) SIGMAR1NPY5RCTSCAVPR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1904477-A1 INDOL-3-CARBONYL-SPIRO-PIPERIDINE DERIVATIVES AS V1A RECEPTOR ANTAGONISTS F. Hoffmann-Roche AG (CH) 2008-04-02 EP disclosed
WO-2007006688-A1 INDOL-3-CARBONYL-SPIRO-PIPERIDINE DERIVATIVES AS V1A RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2007-01-18 WO disclosed