SCHEMBL5136715

SCHEMBL5136715

CCCCn1c(-c2ccccc2)nc(-c2ccccc2)c1CN(Cc1ccccc1)Cc1cccc(OC)c1OC

nearest known ligand 0.43

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
C5AR1 P21730 1/20 0.43
BCHE P06276 16/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
EPHX2 P34913 1/20 0.40
CASR P41180 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5136313 0.95 BCHE (0.43) C5AR1BCHEMEN1KMT2AEPHX2
SCHEMBL5074353 0.93 C5AR1 (0.44) C5AR1BCHEMEN1KMT2ACASR
SCHEMBL5137301 0.92 BCHE (0.45) C5AR1BCHEMEN1KMT2AEPHX2
SCHEMBL5137330 0.92 BCHE (0.43) C5AR1BCHEMEN1KMT2AEPHX2
SCHEMBL5135915 0.88 BCHE (0.41) C5AR1BCHEMEN1KMT2AEPHX2
SCHEMBL5134673 0.87 C5AR1 (0.43) C5AR1BCHECASR
SCHEMBL5137401 0.87 CASR (0.41) C5AR1BCHEMEN1KMT2AEPHX2
SCHEMBL5138021 0.86 C5AR1 (0.43) C5AR1MEN1KMT2ACASR
SCHEMBL5136651 0.85 C5AR1 (0.43) C5AR1MEN1KMT2A
SCHEMBL651094 0.85 TSHR (0.50) C5AR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1490044-A4 COMBINATION THERAPY FOR THE TREATMENT OF CONDITIONS WITH PATHOGENIC INFLAMMATORY COMPONENTS NEUROGEN CORP (US) 2008-04-16 EP disclosed
EP-1490044-A1 COMBINATION THERAPY FOR THE TREATMENT OF CONDITIONS WITH PATHOGENIC INFLAMMATORY COMPONENTS NEUROGEN CORPORATION (US) 2004-12-29 EP disclosed
WO-2003084524-A1 COMBINATION THERAPY FOR THE TREATMENT OF CONDITIONS WITH PATHOGENIC INFLAMMATORY COMPONENTS NEUROGEN CORPORATION (US) 2003-10-16 WO disclosed