SCHEMBL5137301

SCHEMBL5137301

CCCCn1c(-c2ccccc2)nc(-c2ccccc2)c1CN(CCC)Cc1cccc(OC)c1OC

nearest known ligand 0.45

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BCHE P06276 15/20 0.45
C5AR1 P21730 1/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
EPHX2 P34913 1/20 0.41
CASR P41180 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5137330 0.96 BCHE (0.43) BCHEC5AR1MEN1KMT2AEPHX2
SCHEMBL5135193 0.92 BCHE (0.43) BCHEC5AR1CASR
SCHEMBL5135915 0.92 BCHE (0.41) BCHEC5AR1MEN1KMT2AEPHX2
SCHEMBL5136715 0.92 C5AR1 (0.43) BCHEC5AR1MEN1KMT2AEPHX2
SCHEMBL5137401 0.91 CASR (0.41) BCHEC5AR1MEN1KMT2AEPHX2
SCHEMBL5136313 0.89 BCHE (0.43) BCHEC5AR1MEN1KMT2AEPHX2
SCHEMBL5069962 0.89 BCHE (0.45) BCHEC5AR1CASR
SCHEMBL5070121 0.86 SMN1; SMN2 (0.41) BCHEC5AR1
SCHEMBL5135095 0.86 BCHE (0.47) BCHEC5AR1
SCHEMBL5138086 0.86 C5AR1 (0.42) BCHEC5AR1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1490044-A4 COMBINATION THERAPY FOR THE TREATMENT OF CONDITIONS WITH PATHOGENIC INFLAMMATORY COMPONENTS NEUROGEN CORP (US) 2008-04-16 EP disclosed
EP-1490044-A1 COMBINATION THERAPY FOR THE TREATMENT OF CONDITIONS WITH PATHOGENIC INFLAMMATORY COMPONENTS NEUROGEN CORPORATION (US) 2004-12-29 EP disclosed
WO-2003084524-A1 COMBINATION THERAPY FOR THE TREATMENT OF CONDITIONS WITH PATHOGENIC INFLAMMATORY COMPONENTS NEUROGEN CORPORATION (US) 2003-10-16 WO disclosed