SCHEMBL5136738

SCHEMBL5136738

Cc1cc(OCCN2CCC(n3ccnc3)CC2)nn1-c1ccc(Cl)c(Cl)c1

nearest known ligand 0.71

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 20/20 0.71
KCNH2 Q12809 3/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL1897332 0.82 SIGMAR1 (0.98) SIGMAR1KCNH2
SCHEMBL467323 0.81 SIGMAR1 (1.00) SIGMAR1KCNH2
SCHEMBL467171 0.80 SIGMAR1 (1.00) SIGMAR1KCNH2
SCHEMBL466940 0.80 SIGMAR1 (1.00) SIGMAR1KCNH2
SCHEMBL467027 0.80 SIGMAR1 (1.00) SIGMAR1KCNH2
SCHEMBL4560092 0.80 SIGMAR1 (0.78) SIGMAR1KCNH2
SCHEMBL467246 0.80 SIGMAR1 (1.00) SIGMAR1KCNH2
SCHEMBL467159 0.80 SIGMAR1 (0.77) SIGMAR1KCNH2
Hydrochloric Acid SCHEMBL1900361 0.80 SIGMAR1 (0.80) SIGMAR1KCNH2
SCHEMBL19988158 0.79 SIGMAR1 (0.85) SIGMAR1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1994032-A1 PYRAZOLE DERIVATIVES AS SIGMA RECEPTOR INHIBITORS Laboratorios del Dr. Esteve S.A. (ES) 2008-11-26 EP disclosed
WO-2007098953-A1 PYRAZOLE DERIVATIVES AS SIGMA RECEPTOR INHIBITORS LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2007-09-07 WO disclosed