SCHEMBL5137237

SCHEMBL5137237

OC(CN1CCC(Nc2ncnc3[nH]ncc23)CC1)c1ccccc1F

nearest known ligand 0.57

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 13/20 0.57
KCNH2 Q12809 5/20 0.56
CYP2D6 P10635 1/20 0.56
PAK1 Q13153 6/20 0.53
HPGDS O60760 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8256381 1.00 GRIN2B (0.57) GRIN2BKCNH2CYP2D6PAK1HPGDS
SCHEMBL4312440 0.87 GRIN2B (0.57) GRIN2BKCNH2CYP2D6PAK1HPGDS
SCHEMBL14010343 0.82 HPGDS (0.49) GRIN2BKCNH2CYP2D6PAK1HPGDS
SCHEMBL5006285 0.82 HPGDS (0.49) GRIN2BKCNH2CYP2D6PAK1HPGDS
SCHEMBL5006282 0.82 HPGDS (0.49) GRIN2BKCNH2CYP2D6PAK1HPGDS
SCHEMBL5007384 0.82 HPGDS (0.49) GRIN2BKCNH2CYP2D6PAK1HPGDS
SCHEMBL5007376 0.82 HPGDS (0.49) GRIN2BKCNH2CYP2D6PAK1HPGDS
SCHEMBL14010338 0.82 HPGDS (0.49) GRIN2BKCNH2CYP2D6PAK1HPGDS
SCHEMBL4308430 0.81 GRIN2B (0.60) GRIN2BKCNH2CYP2D6PAK1HPGDS
SCHEMBL4317078 0.77 GRIN2B (0.74) GRIN2BKCNH2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874318-A2 N-ALKYL-AZACYCLOALKYL NMDA/NR2B ANTAGONISTS Merck & Co., Inc. (US) 2008-01-09 EP disclosed
WO-2006113471-A2 N-ALKYL-AZACYCLOALKYL NMDA/NR2B ANTAGONISTS MERCK & CO., INC. (US) 2006-10-26 WO disclosed