SCHEMBL5137462

SCHEMBL5137462

C=CNNC(=O)C=C

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25369963 0.81 TSHR (0.53)
SCHEMBL18074609 0.78
SCHEMBL6695144 0.75 TSHR (0.48)
SCHEMBL15224096 0.73
SCHEMBL16809281 0.71
SCHEMBL909232 0.71
SCHEMBL5470839 0.71
SCHEMBL11843098 0.71
SCHEMBL16808897 0.71
SCHEMBL4297899 0.70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730351-A4 COMPOSITION FOR INCREASING CELLULOSIC PRODUCT STRENGTH AND METHOD OF INCREASING CELLULOSIC PRODUCT STRENGTH UNIV PITTSBURGH (US) 2008-03-26 EP claimed
EP-1730351-A2 COMPOSITION FOR INCREASING CELLULOSIC PRODUCT STRENGTH AND METHOD OF INCREASING CELLULOSIC PRODUCT STRENGTH UNIVERSITY OF PITTSBURGH (US) 2006-12-13 EP claimed
EP-1725616-A2 NETWORKED POLYMERIC GELS AND USE OF SUCH POLYMERIC GELS IN HYDROCARBON RECOVERY UNIVERSITY OF PITTSBURGH (US) 2006-11-29 EP claimed
WO-2005089175-A2 COMPOSITION AND METHOD FOR INCREASING CELLULOSIC PRODUCT STRENGTH UNIVERSITY OF PITTSBURGH (US) 2005-09-29 WO claimed
WO-2005085361-A2 NETWORKED POLYMERIC GELS AND USE OF SUCH POLYMERIC GELS IN HYDROCARBON RECOVERY UNIVERSITY OF PITTSBURGH (US) 2005-09-15 WO claimed
US-20050194145-A1 Networked polymeric gels and use of such polymeric gels in hydrocarbon recovery PITTSBURGH, UNIVERSITY OF 2005-09-08 US claimed
EP-1540082-A1 COMPOSITION AND METHOD FOR INCREASING THE STRENGTH OF A CELLULOSIC PRODUCT UNIVERSITY OF PITTSBURGH (US) 2005-06-15 EP claimed
WO-2004025027-A9 COMPOSITION AND METHOD FOR INCREASING THE STRENGTH OF A CELLULOSIC PRODUCT UNIV PITTSBURGH (US) 2004-06-24 WO claimed
WO-2004025027-A1 COMPOSITION AND METHOD FOR INCREASING THE STRENGTH OF A CELLULOSIC PRODUCT UNIVERSITY OF PITTSBURGH (US) 2004-03-25 WO claimed
US-20230219986-A1 NOVEL AMINOPYRIMIDINE EGFR INHIBITOR QILU PHARMACEUTICAL CO., LTD. (CN) 2023-07-13 US disclosed
US-10633348-B2 Methods to treat lymphoplasmacytic lymphoma DANA-FARBER CANCER INSTITUTE, INC. (US) 2020-04-28 US disclosed
US-10597387-B2 Methods to treat lymphoplasmacytic lymphoma DANA-FARBER CANCER INSTITUTE, INC. (US) 2020-03-24 US disclosed
US-20180194739-A1 METHODS TO TREAT LYMPHOPLASMACYTIC LYMPHOMA DANA-FARBER CANCER INSTITUTE, INC. 2018-07-12 US disclosed
US-20180186780-A1 METHODS TO TREAT LYMPHOPLASMACYTIC LYMPHOMA DANA-FARBER CANCER INSTITUTE, INC. (US) 2018-07-05 US disclosed
US-9908872-B2 Methods to treat lymphoplasmacytic lymphoma DANA-FARBER CANCER INSTITUTE, INC. (US) 2018-03-06 US disclosed