SCHEMBL5139969

SCHEMBL5139969

COc1cc2c(NN3C=COC3)ncnc2cc1OCc1cccc(S(=N)(=O)c2cccc(COc3cc4ncnc(NN5C=COC5)c4cc3OC)c2)c1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EGFR P00533 9/20 0.43
LRRK2 Q5S007 4/20 0.43
HTT P42858 4/20 0.43
KDM4E B2RXH2 2/20 0.43
LMNA P02545 1/20 0.43
HPGD P15428 1/20 0.43
LCK P06239 1/20 0.42
GAK O14976 1/20 0.42
MAPK1 P28482 2/20 0.42
RAF1 P04049 1/20 0.42
KDR P35968 3/20 0.41
RET P07949 1/20 0.41
NSD2 O96028 1/20 0.40
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1708350 0.94 LRRK2 (0.42) EGFRLRRK2HTTKDM4ELMNA
SCHEMBL1707947 0.94 LRRK2 (0.43) EGFRLRRK2HTTKDM4ELMNA
SCHEMBL3423878 0.84 EGFR (0.45) EGFRHTTKDM4ELMNAHPGD
SCHEMBL5139968 0.84 HTT (0.42) EGFRHTTKDM4ELMNAHPGD
SCHEMBL5132792 0.77 EGFR (0.50) EGFRLRRK2HTTKDM4ELMNA
SCHEMBL1755275 0.74 NSD2 (0.57) EGFRLRRK2HTTKDM4ELMNA
SCHEMBL1706637 0.73 EGFR (0.50) EGFRLRRK2HTTKDM4ELMNA
SCHEMBL1707567 0.73 NSD2 (0.56) EGFRLRRK2HTTKDM4ELMNA
SCHEMBL1707506 0.73 EGFR (0.49) EGFRLRRK2HTTKDM4ELMNA
SCHEMBL1841010 0.73 NSD2 (0.58) EGFRLRRK2HTTKDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7863283-B2 Sulphoximine-substituted quinazoline derivatives as immuno-modulators, their preparation and use as medicaments BAYER SCHERING PHARMA AG (DE) 2011-01-04 US claimed