SCHEMBL5139968

SCHEMBL5139968

COc1cc2c(NN3C=COC3)ncnc2cc1OCc1cccc(N=[SH2]=O)c1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.42
MAPK1 P28482 2/20 0.42
RAF1 P04049 1/20 0.42
KDR P35968 10/20 0.42
EGFR P00533 7/20 0.42
KDM4E B2RXH2 1/20 0.41
LMNA P02545 1/20 0.41
HPGD P15428 1/20 0.41
LCK P06239 1/20 0.41
GAK O14976 1/20 0.41
EPHA2 P29317 5/20 0.40
EPHB4 P54760 2/20 0.40
FLT1 P17948 1/20 0.40
ERBB2 P04626 2/20 0.40
NSD2 O96028 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5139969 0.84 EGFR (0.43) HTTMAPK1RAF1KDREGFR
SCHEMBL1708350 0.83 LRRK2 (0.42) HTTMAPK1RAF1KDREGFR
SCHEMBL1707947 0.82 LRRK2 (0.43) HTTMAPK1RAF1KDREGFR
SCHEMBL3423878 0.81 EGFR (0.45) HTTMAPK1RAF1KDREGFR
SCHEMBL5132790 0.77 EGFR (0.49) HTTMAPK1RAF1KDREGFR
SCHEMBL30891782 0.64 EGFR (0.83) HTTKDREGFRKDM4ELMNA
SCHEMBL1841010 0.63 NSD2 (0.58) HTTMAPK1RAF1EGFRKDM4E
SCHEMBL1839570 0.62 EGFR (0.51) HTTMAPK1RAF1KDREGFR
SCHEMBL1755275 0.62 NSD2 (0.57) HTTMAPK1RAF1EGFRKDM4E
SCHEMBL1843051 0.62 NSD2 (0.56) HTTMAPK1RAF1EGFRKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7863283-B2 Sulphoximine-substituted quinazoline derivatives as immuno-modulators, their preparation and use as medicaments BAYER SCHERING PHARMA AG (DE) 2011-01-04 US claimed