SCHEMBL5140192

SCHEMBL5140192

CCOc1nc(N)nc2ccc(-c3ccc(C(N)=O)cc3)cc12.Nc1nc(O[C@H]2CCOC2)c2cc(-c3ccc(C(=O)NC4CC4)cc3)ccc2n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BMPR1B O00238 1/20 0.39
BMPR1A P36894 1/20 0.39
TGFBR1 P36897 1/20 0.39
ACVRL1 P37023 1/20 0.39
ACVR1 Q04771 1/20 0.39
F2 P00734 3/20 0.38
F10 P00742 3/20 0.38
PRSS1 P07477 3/20 0.38
PRSS2 P07478 3/20 0.38
F7 P08709 3/20 0.38
F3 P13726 3/20 0.38
PRSS3 P35030 3/20 0.38
MAPK14 Q16539 1/20 0.38
RIPK2 O43353 1/20 0.38
KMT2A Q03164 2/20 0.37
MEN1 O00255 1/20 0.37
RAB9A P51151 1/20 0.37
ATR Q13535 1/20 0.37
HPGDS O60760 1/20 0.37
TYK2 P29597 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3336644 0.91 MEN1 (0.42) MAPK14RIPK2KMT2AMEN1RAB9A
SCHEMBL3336650 0.91 MEN1 (0.42) MAPK14RIPK2KMT2AMEN1RAB9A
SCHEMBL3334673 0.86 MAPK14 (0.47) BMPR1BBMPR1ATGFBR1ACVRL1ACVR1
SCHEMBL3335812 0.83 HRH3 (0.49) TLR7
SCHEMBL3335817 0.83 HRH3 (0.49) TLR7
SCHEMBL3340784 0.83 RAB9A (0.46) BMPR1BBMPR1ATGFBR1ACVRL1ACVR1
SCHEMBL3337545 0.82 RAB9A (0.47) BMPR1BBMPR1ATGFBR1ACVRL1ACVR1
SCHEMBL3335691 0.80 MELK (0.45)
SCHEMBL3335680 0.80 MELK (0.45)
SCHEMBL3341520 0.79 CHEK2 (0.46) PDE4APDE4BPDE4CPDE4DFYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009077-A2 4,6-DL- AND 2,4,6-TRISUBSTITUTED QUINAZOLINE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS USEFUL FOR TREATING VIRAL INFECTIONS GILEAD SCIENCES, INC. (US) 2008-01-24 WO claimed