SCHEMBL514473

SCHEMBL514473

CC(=O)N[C@H](C=O)CS

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16103901 1.00
SCHEMBL13666967 1.00
SCHEMBL13954515 0.83 KDM4E (0.41)
SCHEMBL936834 0.79
SCHEMBL13101176 0.79
SCHEMBL3990275 0.79
SCHEMBL12246397 0.78 KDM4E (0.36)
SCHEMBL24866666 0.77
SCHEMBL3537241 0.77
SCHEMBL23288380 0.77 ALDH1A1 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 47 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109655540-B Method for analyzing related substances of salmon calcitonin nasal spray 银谷制药有限责任公司 2022-08-30 CN claimed
US-7585846-B2 Compounds for delivering amino acids or peptides with antioxidant activity into mitochondria and use thereof UNIVERSITY OF ROCHESTER (US) 2009-09-08 US claimed
US-6335176-B1 REAGENT IS SUCCINIMIDYL MOIETY LINKED TO KINASE SUBSTRATE; CAN BE LINKED TO FREE PRIMARY OR SECONDARY AMINE IN COMPOUND TO BE PHOSPHORYLATED PHARMACOPEIA, INC. 2002-01-01 US claimed
CN-111558049-B Methylene carbamate linkers for use with target-drug conjugates 西雅图基因公司 2024-06-21 CN disclosed
CN-111569086-B Methylene carbamate linkers for use with target-drug conjugates 西雅图基因公司 2024-06-21 CN disclosed
EP-4212181-A2 METHYLENE CARBAMATE LINKERS FOR USE WITH TARGETED-DRUG CONJUGATES Seagen Inc. (US) 2023-07-19 EP disclosed
CN-109655540-B Method for analyzing related substances of salmon calcitonin nasal spray 银谷制药有限责任公司 2022-08-30 CN disclosed
EP-3283461-B1 NOVEL COUMARIN DERIVATIVE FOR DETECTION OF CYSTEINE AND PROCESS FOR THE SYNTHESIS THEREOF COUNCIL SCIENT IND RES (IN) 2022-03-30 EP disclosed
US-20220054650-A1 Methylene Carbamate Linkers for use with Targeted-Drug Conjugates SEATTLE GENETICS, INC. 2022-02-24 US disclosed
US-11116847-B2 Methylene carbamate linkers for use with targeted-drug conjugates SEAGEN INC. (US) 2021-09-14 US disclosed
US-10758498-B2 Method of decreasing protein-aldehyde adducts by administering a mixed disulfide of n-acetylcysteine and propyl mercaptan, propenyl mercaptan, or allyl mercaptan SOCTRONICS TECHNOLOGIES PRIVATE LIMITED (IN) 2020-09-01 US disclosed
WO-2006083692-A2 METHODS OF IDENTIFYING MODULATORS OF BROMODOMAINS MOUNT SINAI SCHOOOL OF MEDICINE (US) 2006-08-10 WO disclosed
US-20030119909-A1 Stabilized medicament containing cysteinyl derivatives STANISLAUS, FRITZ (DE) 2003-06-26 US disclosed
US-20020037855-A1 Stabilized medicament containing cysteinyl derivatives STANISLAUS FRITZ (DE) 2002-03-28 US disclosed
EP-0850924-B1 Aromatic diselenides and selenosulphides for use as antioxidant agents OXIS ISLE OF MAN LTD (GB) 2001-03-14 EP disclosed
US-6040328-A ANTIOXIDANT AGENTS HAVING CYTOPROTECTING ACTIVITY, AND WATER SOLUBLE OXIS INTERNATIONAL S.A. (US) 2000-03-21 US disclosed
US-5973009-A ANTIOXIDANT AND CYTOPROTECTING ACTIVITY OXIS INTERNATIONAL S.A. (US) 1999-10-26 US disclosed
EP-0850924-A1 Aromatic diselenides and selenosulphides for use as antioxidant agents OXIS Isle of Man, Limited (GB) 1998-07-01 EP disclosed
US-5723501-A Pharmaceutical compositions containing 3-IODO-1,2-propanediol having mucolytic activity CARTER-WALLACE, INC. (US) 1998-03-03 US disclosed
US-5066716-A Synthesis of chloroacetyl and bromoacetyl modified peptides for the preparation of synthetic peptide polymers, conjugated peptides, and cyclic peptides THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1991-11-19 US disclosed