SCHEMBL5146366

SCHEMBL5146366

CCN(CC)CCOc1cc2ncnc(Oc3ccc(NC(=O)C4(C(N)=O)CCC4)cc3F)c2cc1OC

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MET P08581 11/20 0.64
KDR P35968 10/20 0.50
AXL P30530 4/20 0.50
FLT3 P36888 4/20 0.49
KIT P10721 3/20 0.49
HDAC2 Q92769 2/20 0.49
HDAC8 Q9BY41 2/20 0.49
HDAC6 Q9UBN7 2/20 0.49
RET P07949 2/20 0.49
PDGFRB P09619 2/20 0.49
HDAC10 Q969S8 1/20 0.48
HDAC11 Q96DB2 1/20 0.48
EGFR P00533 4/20 0.48
AURKA O14965 2/20 0.47
STK10 O94804 2/20 0.47
NTRK1 P04629 2/20 0.47
CDK11B P21127 2/20 0.47
BLK P51451 2/20 0.47
TYRO3 Q06418 2/20 0.47
DDR1 Q08345 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL371698 0.93 MET (0.76) METKDRAXLFLT3KIT
SCHEMBL29693465 0.93 MET (0.76) METKDRAXLFLT3KIT
SCHEMBL19372937 0.90 MET (0.68) METKDRAXLFLT3KIT
SCHEMBL29693470 0.89 MET (0.75) METKDRAXLFLT3KIT
SCHEMBL372151 0.89 MET (0.75) METKDRAXLFLT3KIT
SCHEMBL19373184 0.86 MET (0.68) METKDRAXLFLT3KIT
SCHEMBL371866 0.86 MET (0.79) METKDRAXLFLT3KIT
SCHEMBL19372954 0.86 MET (0.60) METKDRAXLFLT3KIT
SCHEMBL19373004 0.85 MET (0.71) METKDRAXLFLT3KIT
SCHEMBL19372958 0.85 MET (0.64) METKDRAXLFLT3KIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070054928-A1 c-Met modulators and methods of use EXELIXIS, INC. (US) 2007-03-08 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070054928-A1 c-Met modulators and methods of use FLT4, FLT1, MET MET 3/4885KDR 4/4885AXL 109/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.