SCHEMBL5146979

SCHEMBL5146979

COc1ccc2[nH]cc(CCN(CF)C(C)=O)c2c1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.66
HTR1A P08908 6/20 0.64
HTR1D P28221 6/20 0.64
MTNR1A P48039 5/20 0.64
HTR1B P28222 5/20 0.64
CYP2D6 P10635 3/20 0.64
HTR2B P41595 3/20 0.64
MTNR1B P49286 3/20 0.64
CYP1A2 P05177 3/20 0.64
HTR2A P28223 3/20 0.64
HTR2C P28335 3/20 0.64
HTR7 P34969 3/20 0.64
HTR6 P50406 3/20 0.64
HTR1E P28566 2/20 0.64
HTR5A P47898 2/20 0.64
HTR4 Q13639 2/20 0.64
HTR3E A5X5Y0 1/20 0.64
HTR3B O95264 1/20 0.64
CYP2C9 P11712 1/20 0.64
HTR1F P30939 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4075720 0.88 KMT2A (0.72) KMT2AHTR1AHTR1DMTNR1AHTR1B
SCHEMBL5144423 0.84 KMT2A (0.74) KMT2AHTR1AHTR1DMTNR1AHTR1B
SCHEMBL466333 0.84 KMT2A (0.70) KMT2AHTR1AHTR1DMTNR1AHTR1B
SCHEMBL5227242 0.83 KMT2A (0.69) KMT2AHTR1AHTR1DMTNR1AHTR1B
SCHEMBL28414663 0.83 KMT2A (0.69) KMT2AHTR1AHTR1DMTNR1AHTR1B
SCHEMBL16058705 0.83 KMT2A (0.69) KMT2AHTR1AHTR1DMTNR1AHTR1B
SCHEMBL5144364 0.83 KMT2A (0.65) KMT2AHTR1AHTR1DMTNR1AHTR1B
SCHEMBL5085972 0.81 KMT2A (0.65) KMT2AHTR1AHTR1DMTNR1AHTR1B
SCHEMBL5085568 0.81 KMT2A (0.65) KMT2AHTR1AHTR1DMTNR1AHTR1B
Mebufotenin SCHEMBL7205139 0.80 KMT2A (1.00) KMT2AHTR1AHTR1DMTNR1AHTR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1476152-A4 USE OF MELATONIN ANALOGUES FOR INDUCTION OF GENERAL ANESTHESIA UNIV IOWA RES FOUND (US) 2007-04-11 EP disclosed
EP-1476152-A2 USE OF MELATONIN ANALOGUES FOR INDUCTION OF GENERAL ANESTHESIA University of Iowa Research Foundation (US) 2004-11-17 EP disclosed
WO-2003070177-A2 USE OF MELATONIN ANALOGUES FOR INDUCTION OF GENERAL ANESTHESIA UNIVERSITY OF IOWA RESEARCH FOUNDATION (US) 2003-08-28 WO disclosed