SCHEMBL5147702

SCHEMBL5147702

CCCCCCC1=C(N[C@@H](Cc2ccc(Oc3nccc4ccncc34)cc2)C(=O)OCC)C(C)(C)C1=O

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 5/20 0.34
ITGA4 P13612 5/20 0.34
ELANE P08246 1/20 0.33
SLC10A1 Q14973 1/20 0.33
DRD1 P21728 1/20 0.33
PLA2G4A P47712 2/20 0.32
PLG P00747 4/20 0.32
ICAM1 P05362 1/20 0.32
SELE P16581 1/20 0.32
PLAU P00749 1/20 0.32
PRSS1 P07477 1/20 0.32
PRSS2 P07478 1/20 0.32
PRSS3 P35030 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2986901 0.92 ITGB1 (0.41) ITGB1ITGA4SLC10A1
SCHEMBL3873136 0.84 ITGB1 (0.38) ITGB1ITGA4SLC10A1ICAM1SELE
SCHEMBL2987403 0.84 ITGB1 (0.38) ITGB1ITGA4SLC10A1ICAM1SELE
SCHEMBL5147510 0.81 ITGB1 (0.44) ITGB1ITGA4ELANEDRD1
SCHEMBL5147705 0.81 FFAR1 (0.34) SLC10A1DRD1
SCHEMBL3837352 0.80 ITGB1 (0.45) ITGB1ITGA4ELANEDRD1
SCHEMBL5147710 0.79 FFAR1 (0.33) DRD1PLA2G4AICAM1SELE
SCHEMBL7259514 0.79 ITGB1 (0.41) ITGB1ITGA4ELANEDRD1
SCHEMBL7259520 0.79 ITGB1 (0.41) ITGB1ITGA4ELANEDRD1
SCHEMBL5261691 0.79 DRD1 (0.36) ITGB1ITGA4ELANEDRD1PLG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070167483-A1 2-[(2-Isopropylsulfanyl-3-oxo-spiro[3.5]non-1-en-1-yl)amino]-3-[4-([2,7]naphthyridin-1-ylamino)phenyl]propanoic acid; compounds can inhibit the binding of integrins to their ligands and are of use in the prophylaxis and treatment of immuno or inflammatory disorders UCB PHARMA S.A. (BE) 2007-07-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070167483-A1 2-[(2-Isopropylsulfanyl-3-oxo-spiro[3.5]non-1-en-1-yl)amino]-3-[4-([2,7]naphthyridin-1-ylamino)phenyl]propanoic acid; compounds can inhibit the binding of integrins to their ligands and are of use in the prophylaxis and treatment of immuno or inflammatory disorders ITGB2, VCAM1, ITGB1 ITGB1 3/4885ITGA4 40/4885ELANE 275/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.