SCHEMBL5153350

SCHEMBL5153350

CCCSc1cc(C(=O)OC)cc(NC(C)CC)n1.CCC[S+]([O-])c1cc(C(=O)O)cc(NC(C)CC)n1

nearest known ligand 0.34

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 4/20 0.34
CXCR2 P25025 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3855865 0.88 HCAR3 (0.37) HCAR3
SCHEMBL3855868 0.88 HCAR3 (0.37) HCAR3
SCHEMBL3855861 0.88 HCAR3 (0.37) HCAR3
SCHEMBL3854231 0.86 HCAR3 (0.39) HCAR3CXCR2
SCHEMBL3854237 0.86 HCAR3 (0.39) HCAR3CXCR2
SCHEMBL3854435 0.84 HCAR3 (0.45) HCAR3CXCR2
SCHEMBL3862330 0.84 HCAR3 (0.45) HCAR3CXCR2
SCHEMBL3862339 0.84 HCAR3 (0.45) HCAR3CXCR2
SCHEMBL5158231 0.74 CXCR2 (0.33) HCAR3CXCR2
SCHEMBL3854282 0.74 HCAR3 (0.41) HCAR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1740573-A1 AMIDES AS BACE INHIBITORS ELI LILLY AND COMPANY (US) 2007-01-10 EP disclosed
EP-1740575-A2 PYRROLIDINE DERIVATIVES USEFUL AS BACE INHIBITORS ELI LILLY AND COMPANY (US) 2007-01-10 EP disclosed
WO-2005108358-A2 PYRROLIDINE DERIVATIVES USEFUL AS BACE INHIBITORS ELI LILLY AND COMPANY (US) 2005-11-17 WO disclosed
WO-2005108391-A1 AMIDES AS BACE INHIBITORS ELI LILLY AND COMPANY (US) 2005-11-17 WO disclosed