SCHEMBL5158745

SCHEMBL5158745

CC(Oc1ccccc1)C(=O)NC1CCC(Cc2ccccc2)(N2CCCCCC2)CC1.NC(=O)C1CCC(Cc2ccccc2)(N2CCCCCC2)CC1

nearest known ligand 0.55

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.44
SMN1; SMN2 Q16637 3/20 0.39
HPGD P15428 2/20 0.39
CYP2C19 P33261 1/20 0.38
ALDH1A1 P00352 2/20 0.38
KMT2A Q03164 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
RAB9A P51151 2/20 0.37
POLB P06746 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
MAPT P10636 1/20 0.36
HTT P42858 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2989191 0.94 TSHR (0.49) TSHRSMN1; SMN2HPGDCYP2C19ALDH1A1
SCHEMBL2982591 0.93 TSHR (0.50) TSHRSMN1; SMN2HPGDCYP2C19ALDH1A1
SCHEMBL2989357 0.82 TSHR (0.46) TSHRSMN1; SMN2HPGDCYP2C19ALDH1A1
SCHEMBL2989327 0.82 TSHR (0.48) TSHRSMN1; SMN2CYP2C19ALDH1A1KMT2A
SCHEMBL5243972 0.82 TSHR (0.48) TSHRSMN1; SMN2CYP2C19ALDH1A1KMT2A
SCHEMBL4873013 0.81 SMN1; SMN2 (0.47) TSHRSMN1; SMN2CYP2C19ALDH1A1KMT2A
SCHEMBL4867919 0.76 CYP1A2 (0.48) TSHRALDH1A1KMT2AMAPT
SCHEMBL2985459 0.75 POLB (0.59) SMN1; SMN2HPGDCYP2C19ALDH1A1KMT2A
SCHEMBL2983320 0.75 POLB (0.59) SMN1; SMN2HPGDCYP2C19ALDH1A1KMT2A
SCHEMBL2985406 0.75 TSHR (0.54) TSHRSMN1; SMN2HPGDNPSR1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1747191-A1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES WITH A CHAIN EXTENSION Grünenthal GmbH (DE) 2007-01-31 EP disclosed
WO-2005110975-A1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES WITH A CHAIN EXTENSION Grünenthal GmbH (DE) 2005-11-24 WO disclosed