SCHEMBL4867919

SCHEMBL4867919

CC(NC(=O)OCc1ccccc1)C(=O)NC1CCC(Cc2ccccc2)(N2CCCCC2)CC1

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.48
PREP P48147 2/20 0.48
CTSK P43235 7/20 0.46
ELANE P08246 1/20 0.46
CTSL P07711 1/20 0.46
CTSB P07858 1/20 0.46
CYP3A4 P08684 2/20 0.46
TSHR P16473 2/20 0.46
ALDH1A1 P00352 2/20 0.46
MAPT P10636 1/20 0.46
DPP4 P27487 2/20 0.45
KCNH2 Q12809 2/20 0.45
DPP7 Q9UHL4 2/20 0.45
TP53 P04637 1/20 0.45
EPHX1 P07099 1/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4867100 0.88 CYP3A4 (0.49) CYP1A2CTSLCYP3A4TSHRALDH1A1
SCHEMBL4868349 0.83 CTSK (0.51) CTSKCTSLCTSBALDH1A1
SCHEMBL11431644 0.83 ALDH1A1 (0.61) CYP1A2PREPCTSKELANECYP3A4
SCHEMBL4868448 0.82 CYP1A2 (0.50) CYP1A2PREPCTSKELANECTSL
SCHEMBL11436545 0.81 ALDH1A1 (0.59) CYP1A2PREPCTSKELANECTSL
SCHEMBL2982591 0.80 TSHR (0.50) TSHRALDH1A1MAPTKMT2A
Acetic Acid SCHEMBL15194442 0.80 CYP1A2 (0.58) CYP1A2PREPCTSKELANECTSL
SCHEMBL4869157 0.78 CYP1A2 (0.49) CYP1A2PREPCTSKELANECTSL
SCHEMBL4863435 0.78 CYP1A2 (0.46) CYP1A2PREPCTSKCTSLCTSB
SCHEMBL4871937 0.78 SCN9A (0.52) CTSKCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1751090-B1 ACID DERIVATIVES OF SUBSTITUTED CYCLOHEXYL-1,4-DIAMINES GRUENENTHAL GMBH (DE) 2014-10-08 EP claimed
US-7439394-B2 Cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2008-10-21 US claimed
US-20070117803-A1 Cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2007-05-24 US claimed
US-7439394-B2 Cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2008-10-21 US disclosed
US-20070117803-A1 Cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2007-05-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070117803-A1 Cyclohexyl-1,4-diamine compounds PKD1, DDC, DPYD CYP1A2 332/4885PREP 142/4885CTSK 1123/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.