SCHEMBL5160638

SCHEMBL5160638

O=C(O)C(O)(c1ccccc1)c1ccccc1C1CCCNC1

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 1/20 0.41
CHUK O15111 1/20 0.41
CSF1R P07333 1/20 0.41
BTK Q06187 1/20 0.41
HTR6 P50406 2/20 0.40
CYP2C9 P11712 1/20 0.39
KEAP1 Q14145 1/20 0.38
NFE2L2 Q16236 1/20 0.38
JAK3 P52333 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Benzylic Acid SCHEMBL6434928 0.75 CYP2C9 (0.55) CYP2C9KEAP1NFE2L2
SCHEMBL17294705 0.75 ATM (0.50)
SCHEMBL30128750 0.75 ATM (0.50)
SCHEMBL17300855 0.75 HTR2C (0.45) HTR6
SCHEMBL15935173 0.75 HTR2C (0.45) HTR6
SCHEMBL17300856 0.75 HTR2C (0.45) HTR6
SCHEMBL16455234 0.75 HTR2C (0.66) HTR6
Benzylic Acid SCHEMBL27825208 0.74 CYP2C9 (0.53) CYP2C9KEAP1NFE2L2
SCHEMBL1004280 0.74 CHRM3 (0.54) HTR6CYP2C9
Hydrochloric Acid SCHEMBL16446229 0.74 HTR2C (0.67) HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-11152270-A None JP disclosed
EP-1275645-B1 LABELED COMPOUNDS FOR MEASURING THE FUNCTION OF THE MUSCARINIC ACETYLCHOLINE NERVOUS SYSTEM HAMAMATSU PHOTONICS KK (JP) 2007-02-28 EP disclosed
EP-1275645-A1 LABELED COMPOUNDS FOR MEASURING THE FUNCTION OF THE MUSCARINIC ACETYLCHOLINE NERVOUS SYSTEM HAMAMATSU PHOTONICS K. K. (JP) 2003-01-15 EP disclosed
JP-H11152270-A MUSCARINIC ACETYLCHOLINE NERVOUS SYSTEM LABELED COMPOUND AND ITS SYNTHESIS HAMAMATSU PHOTONICS KK 1999-06-08 JP disclosed