SCHEMBL5160905

SCHEMBL5160905

CCN(CCNC(=O)CCC(=O)NC1CCC(c2ccccc2)(N(C)C)CC1)c1cccc(C)c1.NC(=O)c1cccc(Oc2ccccc2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 4/20 0.42
OPRL1 P41146 4/20 0.42
GFER P55789 2/20 0.40
NPC1 O15118 1/20 0.39
PKM P14618 1/20 0.38
NPSR1 Q6W5P4 3/20 0.37
GAA P10253 1/20 0.37
MAPT P10636 7/20 0.37
LMNA P02545 3/20 0.37
ALDH1A1 P00352 3/20 0.37
HPGD P15428 2/20 0.37
TSHR P16473 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
HTT P42858 3/20 0.36
ALOX15 P16050 1/20 0.36
USP2 O75604 1/20 0.36
TP53 P04637 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL206795 0.90 OPRM1 (0.52) OPRM1OPRL1GFERNPSR1GAA
SCHEMBL206667 0.78 NPSR1 (0.42) GFERNPSR1GAAMAPTLMNA
SCHEMBL206791 0.70 OPRM1 (0.62) OPRM1OPRL1HPGD
SCHEMBL207976 0.69 OPRM1 (0.60) OPRM1OPRL1TP53
SCHEMBL207397 0.68 OPRM1 (0.56) OPRM1OPRL1NPSR1MAPTALDH1A1
SCHEMBL208501 0.67 OPRM1 (0.60) OPRM1OPRL1NPC1ALDH1A1HPGD
SCHEMBL207055 0.67 OPRM1 (0.57) OPRM1OPRL1NPSR1HTT
SCHEMBL11661392 0.67 GFER (0.75) GFERNPC1GAAMAPTLMNA
SCHEMBL2974572 0.66 OPRM1 (0.64) OPRM1OPRL1MAPTSMN1; SMN2KMT2A
SCHEMBL9060635 0.66 GFER (0.57) GFERNPC1NPSR1GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007536323-A 2007-12-13 JP claimed
EP-1745010-A1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES Grünenthal GmbH (DE) 2007-01-24 EP claimed
WO-2005110974-A1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES Grünenthal GmbH (DE) 2005-11-24 WO claimed