SCHEMBL5161052

SCHEMBL5161052

CCNC(=O)CC(=O)c1ccncc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLOD2 O00469 3/20 0.56
PLOD3 O60568 3/20 0.56
PLOD1 Q02809 3/20 0.56
ALDH1A1 P00352 3/20 0.56
CYP1A2 P05177 2/20 0.56
CYP3A4 P08684 2/20 0.56
CYP2D6 P10635 2/20 0.56
CYP2C19 P33261 2/20 0.56
CYP2C9 P11712 1/20 0.56
HPGD P15428 1/20 0.56
HIF1A Q16665 1/20 0.56
GAA P10253 2/20 0.53
CA1 P00915 1/20 0.53
CA9 Q16790 1/20 0.53
KMT2A Q03164 2/20 0.47
NAAA Q02083 1/20 0.46
KDM4E B2RXH2 1/20 0.46
MPO P05164 1/20 0.46
ADORA3 P0DMS8 1/20 0.46
CYP2A6 P11509 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7160200 0.88 CYP2D6 (0.45) PLOD2PLOD3PLOD1ALDH1A1CYP1A2
SCHEMBL5160670 0.81 PLOD2 (0.60) PLOD2PLOD3PLOD1ALDH1A1CYP1A2
SCHEMBL10606188 0.81 KMT2A (0.61) PLOD2PLOD3PLOD1ALDH1A1CYP1A2
SCHEMBL5163201 0.80 PLOD2 (0.63) PLOD2PLOD3PLOD1ALDH1A1CYP1A2
SCHEMBL10948430 0.80 PLOD2 (0.83) PLOD2PLOD3PLOD1ALDH1A1CYP1A2
SCHEMBL1028171 0.79 GAA (0.67) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL5164294 0.78 HCAR2 (0.42) PLOD2ALDH1A1GAACA1CA9
SCHEMBL2008122 0.77 CYP1A2 (0.64) PLOD2PLOD3PLOD1ALDH1A1CYP1A2
SCHEMBL27908332 0.76 PLOD2 (0.55) PLOD2PLOD3PLOD1ALDH1A1CYP1A2
SCHEMBL3108729 0.76 PLOD2 (0.64) PLOD2PLOD3PLOD1ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1340746-B1 Process for the reduction of 3-heteroaryl-3-oxo-propanoic acid derivatives SALTIGO GMBH (DE) 2007-02-28 EP disclosed
EP-1340746-A1 Process for the reduction of 3-heteroaryl-3-oxo-propanoic acid derivatives BAYER AG (DE) 2003-09-03 EP disclosed