SCHEMBL5162050

SCHEMBL5162050

CCOC(=O)OC1CCN(C2CCN(C(=O)[C@@H](Cc3cc(C)c(OCc4ccccc4)c(C)c3)OC(=O)N3CCC(N4CCc5ccccc5NC4=O)CC3)CC2)CC1

nearest known ligand 0.65

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CALCRL Q16602 20/20 0.65
RAMP1 O60894 2/20 0.65
CYP3A4 P08684 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4594481 0.94 CALCRL (0.68) CALCRLRAMP1CYP3A4
SCHEMBL2086399 0.92 CALCRL (0.63) CALCRLRAMP1CYP3A4
SCHEMBL2087350 0.91 CALCRL (0.66) CALCRLRAMP1CYP3A4
SCHEMBL5164207 0.91 CALCRL (0.78) CALCRLRAMP1CYP3A4
SCHEMBL2087418 0.90 CALCRL (0.69) CALCRLRAMP1CYP3A4
SCHEMBL10024353 0.89 CALCRL (0.82) CALCRLRAMP1CYP3A4
SCHEMBL2088624 0.88 CALCRL (0.64) CALCRLRAMP1CYP3A4
SCHEMBL2088625 0.88 CALCRL (0.64) CALCRLRAMP1CYP3A4
SCHEMBL2087682 0.87 CALCRL (0.68) CALCRLRAMP1CYP3A4
SCHEMBL2085873 0.87 CALCRL (0.62) CALCRLRAMP1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1770086-A1 Selected CGRP antagonists, process for their preparation as well as their use as medicaments Boehringer Ingelheim Pharma GmbH & Co. KG (DE) 2007-04-04 EP disclosed