SCHEMBL5164207

SCHEMBL5164207

CCOC(=O)OC1CCN(C2CCN(C(=O)[C@@H](Cc3cc(C)c(O)c(C)c3)OC(=O)N3CCC(N4CCc5ccccc5NC4=O)CC3)CC2)CC1

nearest known ligand 0.78

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CALCRL Q16602 20/20 0.78
RAMP1 O60894 2/20 0.78
CYP3A4 P08684 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12773080 0.93 CALCRL (0.81) CALCRLRAMP1CYP3A4
SCHEMBL5165549 0.93 CALCRL (0.81) CALCRLRAMP1CYP3A4
SCHEMBL5162050 0.91 CALCRL (0.65) CALCRLRAMP1CYP3A4
SCHEMBL2085601 0.91 CALCRL (0.83) CALCRLRAMP1CYP3A4
SCHEMBL2088312 0.91 CALCRL (0.76) CALCRLRAMP1CYP3A4
SCHEMBL2086519 0.91 CALCRL (0.80) CALCRLRAMP1CYP3A4
SCHEMBL2086814 0.90 CALCRL (0.86) CALCRLRAMP1CYP3A4
SCHEMBL12773023 0.90 CALCRL (0.89) CALCRLRAMP1CYP3A4
SCHEMBL13712911 0.90 CALCRL (0.71) CALCRLRAMP1CYP3A4
SCHEMBL14016390 0.90 CALCRL (0.88) CALCRLRAMP1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1770086-A1 Selected CGRP antagonists, process for their preparation as well as their use as medicaments Boehringer Ingelheim Pharma GmbH & Co. KG (DE) 2007-04-04 EP disclosed