SCHEMBL5162478

SCHEMBL5162478

CC(C)C(C(=O)O)C(=O)c1ncccn1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.36
CTNNB1 P35222 1/20 0.35
WNT3A P56704 1/20 0.35
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
HSPA5 P11021 1/20 0.34
PTPRA P18433 1/20 0.33
POLB P06746 1/20 0.33
LMNA P02545 2/20 0.33
GSK3B P49841 1/20 0.32
NAPRT Q6XQN6 1/20 0.32
P4HTM Q9NXG6 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
FFAR2 O15552 1/20 0.32
MEN1 O00255 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
KMT2A Q03164 1/20 0.32
ALDH1A1 P00352 3/20 0.31
KDM4E B2RXH2 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5160980 0.79 P2RX7 (0.39) P2RX7CTNNB1WNT3ACYP1A2CYP3A4
SCHEMBL5163592 0.78 GSK3B (0.56) CYP1A2CYP3A4POLBLMNAGSK3B
SCHEMBL13820572 0.76 P2RX7 (0.43) P2RX7CTNNB1WNT3ACYP1A2CYP3A4
SCHEMBL15936878 0.74 P2RX7 (0.41) P2RX7CTNNB1WNT3ACYP1A2CYP3A4
SCHEMBL15936872 0.72 GSK3B (0.44) P2RX7CTNNB1WNT3ACYP1A2CYP3A4
SCHEMBL5162794 0.72 P2RX7 (0.41) P2RX7CTNNB1WNT3ACYP1A2PTPRA
SCHEMBL7021730 0.71 CA12 (0.49) CYP3A4LMNANAPRTL3MBTL1NPC1
SCHEMBL5162688 0.71 NAPRT (0.48) CYP1A2CYP3A4LMNANAPRTMEN1
SCHEMBL24663483 0.69 P2RX7 (0.42) P2RX7CTNNB1WNT3ACYP1A2CYP3A4
SCHEMBL28393062 0.69 P2RX7 (0.42) P2RX7CTNNB1WNT3ACYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1340746-B1 Process for the reduction of 3-heteroaryl-3-oxo-propanoic acid derivatives SALTIGO GMBH (DE) 2007-02-28 EP disclosed
EP-1340746-A1 Process for the reduction of 3-heteroaryl-3-oxo-propanoic acid derivatives BAYER AG (DE) 2003-09-03 EP disclosed