SCHEMBL5163933

SCHEMBL5163933

O=C(CO)Cc1ccc(F)cc1

nearest known ligand 0.59

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.52
CTBP2 P56545 1/20 0.50
TDP1 Q9NUW8 2/20 0.47
POLB P06746 2/20 0.47
APEX1 P27695 1/20 0.47
IDO1 P14902 1/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
ALDH1A1 P00352 1/20 0.46
RAB9A P51151 1/20 0.46
EGFR P00533 1/20 0.46
ERBB2 P04626 1/20 0.46
LMNA P02545 2/20 0.44
HTT P42858 2/20 0.44
KMT2A Q03164 2/20 0.44
KDM4E B2RXH2 1/20 0.44
VNN1 O95497 1/20 0.44
TRPA1 O75762 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL526194 0.88 GAA (0.57) GAACTBP2TDP1POLBAPEX1
SCHEMBL27675295 0.82 GAA (0.52) GAACTBP2TDP1POLBAPEX1
SCHEMBL28221360 0.82 GAA (0.52) GAACTBP2TDP1POLBAPEX1
SCHEMBL17585418 0.81 TSHR (0.42) GAATDP1LMNAHTT
SCHEMBL756910 0.80 PTPN1 (0.52) GAACTBP2TDP1POLBAPEX1
SCHEMBL4641892 0.80 GAA (0.50) GAACTBP2TDP1POLBAPEX1
SCHEMBL14609496 0.80 GAA (0.50) GAACTBP2TDP1POLBAPEX1
SCHEMBL1151049 0.80 GAA (0.50) GAACTBP2TDP1POLBAPEX1
SCHEMBL7256741 0.80 TDP1 (0.55) GAACTBP2TDP1POLBAPEX1
SCHEMBL823410 0.80 GAA (0.50) GAACTBP2TDP1POLBAPEX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1765793-A1 CETP INHIBITORS Merck and Co., Inc. (US) 2007-03-28 EP disclosed
WO-2006014413-A1 CETP INHIBITORS MERCK & CO., INC. (US) 2006-02-09 WO disclosed