SCHEMBL5164091

SCHEMBL5164091

COC(=O)[C@H](Cc1ccc(-c2cn(C)c(=O)n(C)c2=O)c(C)c1)NC(=O)c1c(C)cccc1Cl

nearest known ligand 0.84

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 20/20 0.84
ITGA4 P13612 20/20 0.84
ITGB7 P26010 16/20 0.78
ITGA2 P17301 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5159923 0.97 ITGA4 (0.84) ITGB1ITGA4ITGB7
SCHEMBL5160269 0.91 ITGB1 (1.00) ITGB1ITGA4ITGB7ITGA2
SCHEMBL5160231 0.90 ITGA4 (0.68) ITGB1ITGA4ITGB7
SCHEMBL5161994 0.88 ITGA4 (1.00) ITGB1ITGA4ITGB7
SCHEMBL5165005 0.83 ITGB1 (0.84) ITGB1ITGA4ITGB7
SCHEMBL27494297 0.83 ITGB1 (0.86) ITGB1ITGA4ITGB7
SCHEMBL27494296 0.83 ITGB1 (0.86) ITGB1ITGA4ITGB7
SCHEMBL5164939 0.81 ITGA4 (0.81) ITGB1ITGA4ITGB7ITGA2
SCHEMBL5162949 0.80 ITGA4 (0.59) ITGB1ITGA4ITGB7
SCHEMBL6235244 0.79 ITGA4 (0.64) ITGB1ITGA4ITGB7ITGA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1237878-B1 4-PYRIMIDINYL-N-ACYL-L-PHENYLALANINES HOFFMANN LA ROCHE (CH) 2007-03-21 EP disclosed
EP-1237878-B1 4-PYRIMIDINYL-N-ACYL-L-PHENYLALANINES HOFFMANN LA ROCHE (CH) 2007-03-21 EP disclosed
EP-1237878-A2 4-PYRIMIDINYL-N-ACYL-L-PHENYLALANINES F. HOFFMANN-LA ROCHE AG (CH) 2002-09-11 EP disclosed
US-6380387-B1 ANTIINFLAMMATORY AGENTS, ANTIASTHMATICS HOFFMANN-LA ROCHE INC. 2002-04-30 US disclosed
WO-2001042225-A2 4-PYRIMIDINYL-N-ACYL-L-PHENYLALANINES F. HOFFMANN-LA ROCHE AG (CH) 2001-06-14 WO disclosed