SCHEMBL5165033

SCHEMBL5165033

CN(C)C(=O)Oc1ccc(C[C@H](NC(=O)[C@@H]2CCCN2S(=O)(=O)c2cc(Cl)sc2Cl)C(=O)O)cc1.COc1ccc(S(=O)(=O)N2CCC[C@H]2C(=O)N[C@@H](Cc2ccc(OC(=O)N(C)C)cc2)C(=O)O)cc1

nearest known ligand 0.53

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 4/20 0.53
ITGA4 P13612 3/20 0.53
ITGB7 P26010 1/20 0.53
ITGA5 P08648 2/20 0.47
HCRTR1 O43613 14/20 0.46
HCRTR2 O43614 14/20 0.46
CYP3A4 P08684 2/20 0.44
USP2 O75604 1/20 0.43
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3856977 0.94 ITGB1 (0.55) ITGB1ITGA4ITGB7ITGA5
SCHEMBL3848928 0.90 ITGB1 (0.57) ITGB1ITGA4ITGB7ITGA5HCRTR1
SCHEMBL3852834 0.86 ITGB1 (0.46) ITGB1ITGA4ITGB7ITGA5
SCHEMBL3852610 0.84 ITGA4 (0.61) ITGB1ITGA4ITGB7ITGA5HCRTR1
SCHEMBL3848324 0.83 ITGB1 (0.57) ITGB1ITGA4ITGB7ITGA5HCRTR1
SCHEMBL3855807 0.83 ITGB1 (0.56) ITGB1ITGA4ITGB7ITGA5ALDH1A1
SCHEMBL3851029 0.82 ITGB1 (0.59) ITGB1ITGA4ITGB7ITGA5HCRTR1
SCHEMBL3851032 0.82 ITGB1 (0.59) ITGB1ITGA4ITGB7ITGA5HCRTR1
SCHEMBL7326216 0.82 ITGB1 (0.49) ITGB1ITGA4ITGB7ITGA5
SCHEMBL3850912 0.82 ITGB1 (0.56) ITGB1ITGA4ITGB7ITGA5ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1763361-A2 STEROID SPARING AGENTS AND THEIR USE Elan Pharmaceuticals, Inc. (US) 2007-03-21 EP disclosed
WO-2005097162-A2 STEROID SPARING AGENTS AND THEIR USE ELAN PHARMACEUTICALS, INC. (US) 2005-10-20 WO disclosed