SCHEMBL516574

SCHEMBL516574

FC(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)[S]

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.34
TSHR P16473 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
CYP1A2 P05177 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
RECQL P46063 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16687343 0.84 TSHR (0.42) KDM4ETSHRTDP1CYP1A2CYP2C9
SCHEMBL1825532 0.84 TSHR (0.42) KDM4ETSHRTDP1CYP1A2CYP2C9
SCHEMBL1829371 0.84 TSHR (0.42) KDM4ETSHRTDP1CYP1A2CYP2C9
SCHEMBL5489726 0.84 TSHR (0.42) KDM4ETSHRTDP1CYP1A2CYP2C9
SCHEMBL1824897 0.84 TSHR (0.42) KDM4ETSHRTDP1CYP1A2CYP2C9
SCHEMBL5492824 0.84 TSHR (0.42) KDM4ETSHRTDP1CYP1A2CYP2C9
SCHEMBL1824498 0.84 TSHR (0.42) KDM4ETSHRTDP1CYP1A2CYP2C9
SCHEMBL1827978 0.84 TSHR (0.42) KDM4ETSHRTDP1CYP1A2CYP2C9
SCHEMBL5487202 0.84 TSHR (0.42) KDM4ETSHRTDP1CYP1A2CYP2C9
Water SCHEMBL10544296 0.81 TSHR (0.40) KDM4ETSHRTDP1CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 491 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4396163-A1 HERBICIDAL MALONAMIDES CONTAINING MONOCYCLIC HETEROAROMATIC RINGS BASF SE (DE) 2024-07-10 EP disclosed
EP-4396173-A1 HERBICIDAL MALONAMIDES CONTAINING A CONDENSED RING SYSTEM BASF SE (DE) 2024-07-10 EP disclosed
EP-4392403-A1 HERBICIDAL MALONAMIDES BASF SE (DE) 2024-07-03 EP disclosed
EP-4391808-A1 HERBICIDAL MALONAMIDES BASF SE (DE) 2024-07-03 EP disclosed
CN-117881667-A Herbicide malonamides containing a condensed ring system 巴斯夫欧洲公司 2024-04-12 CN disclosed
CN-117881662-A Herbicide malonamide containing monocyclic heteroaromatic ring 巴斯夫欧洲公司 2024-04-12 CN disclosed
CN-117881656-A Herbicide malonamide 巴斯夫欧洲公司 2024-04-12 CN disclosed
CN-117858619-A Herbicide malonamide 巴斯夫欧洲公司 2024-04-09 CN disclosed
WO-2023031199-A1 HERBICIDAL MALONAMIDES CONTAINING MONOCYCLIC HETEROAROMATIC RINGS BASF SE (DE) 2023-03-09 WO disclosed
WO-2023031200-A1 HERBICIDAL MALONAMIDES CONTAINING A CONDENSED RING SYSTEM BASF SE (DE) 2023-03-09 WO disclosed
WO-2000034270-A1 THIOCHROMANOYLPYRAZOLONE DERIVATIVES BASF AKTIENGESELLSCHAFT (DE) 2000-06-15 WO disclosed
EP-0998472-A1 SUBSTITUTED 2-(BENZOARYL)PYRIDINES BASF AKTIENGESELLSCHAFT (DE) 2000-05-10 EP disclosed
WO-2000014069-A1 CYCLOHEXENONQUINOLINOYL-DERIVATIVES AS HERBICIDAL AGENTS BASF AKTIENGESELLSCHAFT (DE) 2000-03-16 WO disclosed
WO-1999059991-A1 PYRAZOLYLDIOXOTHIOCHROMANOYL DERIVATIVES BASF AKTIENGESELLSCHAFT (DE) 1999-11-25 WO disclosed
EP-0958292-A1 4-(3-HETEROCYCLYL-1-BENZOYL)PYRAZOLES AND THEIR USE AS HERBICIDES BASF AKTIENGESELLSCHAFT (DE) 1999-11-24 EP disclosed
EP-0958291-A1 3-HETEROCYCLYL-SUBSTITUTED BENZOYL DERIVATIVES BASF AKTIENGESELLSCHAFT (DE) 1999-11-24 EP disclosed
WO-1999057111-A1 CYCLOHEXENONDIOXOTHIO CHROMANOYL DERIVATIVES BASF AKTIENGESELLSCHAFT (DE) 1999-11-11 WO disclosed
WO-1999006394-A1 SUBSTITUTED 2-(BENZOARYL)PYRIDINES BASF AKTIENGESELLSCHAFT (DE) 1999-02-11 WO disclosed
WO-1998031681-A1 3-HETEROCYCLYL-SUBSTITUTED BENZOYL DERIVATIVES BASF AKTIENGESELLSCHAFT (DE) 1998-07-23 WO disclosed
WO-1998031682-A1 4-(3-HETEROCYCLYL-1-BENZOYL)PYRAZOLES AND THEIR USE AS HERBICIDES BASF AKTIENGESELLSCHAFT (DE) 1998-07-23 WO disclosed