SCHEMBL5166771

SCHEMBL5166771

COc1ccc(CN2CCCC(O)(c3cccc(OC)c3)C2)cc1

nearest known ligand 0.60

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.60
KDM4E B2RXH2 2/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
CYP3A4 P08684 2/20 0.47
CYP2D6 P10635 2/20 0.47
SIGMAR1 Q99720 6/20 0.47
KMT2A Q03164 3/20 0.47
OPRM1 P35372 1/20 0.47
OPRD1 P41143 1/20 0.47
OPRK1 P41145 1/20 0.47
OPRL1 P41146 1/20 0.47
PTGIR P43119 1/20 0.45
MEN1 O00255 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
CYP1A2 P05177 1/20 0.44
HPGD P15428 1/20 0.44
TSHR P16473 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3098400 0.99 ALDH1A1 (0.59) ALDH1A1KDM4EL3MBTL1CYP3A4CYP2D6
SCHEMBL5166618 0.93 ALDH1A1 (0.58) ALDH1A1KDM4EL3MBTL1SIGMAR1KMT2A
SCHEMBL3081018 0.93 ALDH1A1 (0.60) ALDH1A1KDM4EL3MBTL1CYP3A4CYP2D6
SCHEMBL5168369 0.92 ALDH1A1 (0.57) ALDH1A1KDM4EL3MBTL1SIGMAR1KMT2A
Hydrochloric Acid SCHEMBL3074059 0.92 ALDH1A1 (0.57) ALDH1A1KDM4EL3MBTL1SIGMAR1KMT2A
SCHEMBL5168339 0.92 ALDH1A1 (0.57) ALDH1A1KDM4EL3MBTL1SIGMAR1KMT2A
Hydrochloric Acid SCHEMBL11194779 0.92 ALDH1A1 (0.59) ALDH1A1KDM4EL3MBTL1CYP3A4CYP2D6
Hydrochloric Acid SCHEMBL3074049 0.91 ALDH1A1 (0.56) ALDH1A1KDM4EL3MBTL1SIGMAR1KMT2A
Hydrochloric Acid SCHEMBL3086710 0.91 ALDH1A1 (0.56) ALDH1A1KDM4EL3MBTL1SIGMAR1KMT2A
SCHEMBL5166997 0.90 ALDH1A1 (0.55) ALDH1A1KDM4EL3MBTL1SIGMAR1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1771417-A1 SUBSTITUTED 3-PHENYLPIPERIDINE DERIVATIVES Grünenthal GmbH (DE) 2007-04-11 EP claimed
WO-2006010577-A1 SUBSTITUTED 3-PHENYLPIPERIDINE DERIVATIVES Grünenthal GmbH (DE) 2006-02-02 WO claimed
EP-1771417-A1 SUBSTITUTED 3-PHENYLPIPERIDINE DERIVATIVES Grünenthal GmbH (DE) 2007-04-11 EP disclosed
WO-2006010577-A1 SUBSTITUTED 3-PHENYLPIPERIDINE DERIVATIVES Grünenthal GmbH (DE) 2006-02-02 WO disclosed