SCHEMBL5167050

SCHEMBL5167050

COc1c(N2CC(C)NC(C)C2)c(F)cc2c(=O)c(OC(=O)NCc3ccc(Cl)cc3Cl)cn(CCF)c12

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 4/20 0.41
TOP1 P11387 9/20 0.40
KCNH2 Q12809 2/20 0.39
POLB P06746 2/20 0.39
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 2/20 0.39
TDP1 Q9NUW8 2/20 0.39
PRKD3 O94806 1/20 0.39
HPGD P15428 1/20 0.39
ALOX15 P16050 1/20 0.39
OPRM1 P35372 1/20 0.39
CLK2 P49760 1/20 0.39
HSD17B10 Q99714 1/20 0.39
CLK4 Q9HAZ1 1/20 0.39
LMNA P02545 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5276465 0.92 P2RX7 (0.40) P2RX7TOP1KCNH2POLBKDM4E
SCHEMBL12917322 0.90 TOP1 (0.47) P2RX7TOP1KCNH2POLBKDM4E
SCHEMBL964967 0.90 TOP1 (0.47) P2RX7TOP1KCNH2POLBKDM4E
SCHEMBL5242516 0.89 KDM4E (0.51) KCNH2POLBKDM4EALDH1A1TDP1
SCHEMBL5284756 0.88 KDM4E (0.41) P2RX7TOP1KCNH2POLBKDM4E
SCHEMBL12917323 0.84 TOP1 (0.45) P2RX7TOP1KCNH2POLBKDM4E
SCHEMBL4252792 0.83 TOP1 (0.46) TOP1KCNH2POLBKDM4EALDH1A1
SCHEMBL12917330 0.82 TOP1 (0.45) P2RX7TOP1KCNH2POLBKDM4E
SCHEMBL5283636 0.82 POLB (0.43) P2RX7KCNH2POLBKDM4EALDH1A1
SCHEMBL5182149 0.82 TOP1 (0.39) P2RX7TOP1KCNH2POLBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1768973-B1 SUBSTITUTED QUINOLONES AICURIS GMBH & CO KG (DE) 2007-12-05 EP disclosed
EP-1768973-A1 SUBSTITUTED QUINOLONES AiCuris GmbH & Co. KG (DE) 2007-04-04 EP disclosed
WO-2006008046-A1 SUBSTITUTED QUINOLONES AICURIS GMBH & CO. KG (DE) 2006-01-26 WO disclosed