SCHEMBL5170168

SCHEMBL5170168

O=C(O)/C=C/c1ccc(NC2CCCN(CC3CCCCC3)C2)nc1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 2/20 0.41
ADORA3 P0DMS8 1/20 0.40
ADORA2A P29274 1/20 0.40
ADORA2B P29275 1/20 0.40
ADORA1 P30542 1/20 0.40
KDM2B Q8NHM5 1/20 0.40
CCR1 P32246 1/20 0.39
CHRM2 P08172 4/20 0.39
CHRM4 P08173 4/20 0.39
CHRM5 P08912 4/20 0.39
CHRM1 P11229 4/20 0.39
CHRM3 P20309 4/20 0.39
RARB P10826 1/20 0.39
P4HTM Q9NXG6 1/20 0.38
JAK2 O60674 2/20 0.37
JAK3 P52333 2/20 0.37
CCR2 P41597 1/20 0.37
KCNH2 Q12809 1/20 0.37
PIM2 Q9P1W9 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4215495 1.00 HCAR3 (0.41) HCAR3ADORA3ADORA2AADORA2BADORA1
SCHEMBL4227644 1.00 HCAR3 (0.41) HCAR3ADORA3ADORA2AADORA2BADORA1
SCHEMBL4227640 1.00 HCAR3 (0.41) HCAR3ADORA3ADORA2AADORA2BADORA1
SCHEMBL4215489 1.00 HCAR3 (0.41) HCAR3ADORA3ADORA2AADORA2BADORA1
SCHEMBL4217456 0.90 HDAC1 (0.47) KCNH2
SCHEMBL4217447 0.90 HDAC1 (0.47) KCNH2
SCHEMBL4221891 0.89 P4HTM (0.41) HCAR3KDM2BCCR1P4HTMPIM2
SCHEMBL5168703 0.89 P4HTM (0.41) HCAR3KDM2BCCR1P4HTMPIM2
SCHEMBL4221889 0.89 P4HTM (0.41) HCAR3KDM2BCCR1P4HTMPIM2
Hydrochloric Acid SCHEMBL4223910 0.89 HDAC1 (0.46) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1776357-A1 HYDROXYAMIDE COMPOUNDS HAVING ACTIVITY AS INHIBITORS OF HISTONE DEACETYLASE (HDAC) Astellas Pharma Inc. (JP) 2007-04-25 EP disclosed
WO-2006016680-A1 HYDROXYAMIDE COMPOUNDS HAVING ACTIVITY AS INHIBITORS OF HISTONE DEACETYLASE (HDAC) ASTELLAS PHARMA INC. (JP) 2006-02-16 WO disclosed