SCHEMBL51754

SCHEMBL51754

Cc1ccc([CH]Cc2cccc(C)c2)cc1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 2/20 0.46
ACHE P22303 2/20 0.46
IDO1 P14902 2/20 0.44
MAOB P27338 3/20 0.44
MAOA P21397 2/20 0.44
NFE2L2 Q16236 2/20 0.42
CYP2A6 P11509 1/20 0.40
RELA Q04206 1/20 0.40
TP53 P04637 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
KDM4E B2RXH2 1/20 0.39
HPGD P15428 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
NPC1 O15118 1/20 0.38
CASP3 P42574 1/20 0.38
SENP8 Q96LD8 1/20 0.38
SENP7 Q9BQF6 1/20 0.38
SENP6 Q9GZR1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8097032 0.86 TP53 (0.50) TAAR1ACHEIDO1MAOBMAOA
SCHEMBL1078091 0.84 PNMT (0.44) TAAR1IDO1TP53KDM4E
SCHEMBL1987774 0.82 MAOB (0.46) ACHEMAOBCYP2A6TDP1KDM4E
SCHEMBL4953933 0.81 TP53 (0.48) TAAR1ACHEIDO1MAOBMAOA
SCHEMBL5056468 0.79 CYP2A6 (0.50) TAAR1ACHEIDO1MAOBMAOA
SCHEMBL21179476 0.77 CYP2A6 (0.48) TAAR1ACHEIDO1MAOBMAOA
SCHEMBL8207446 0.77 TP53 (0.48) TAAR1ACHEIDO1MAOBMAOA
SCHEMBL9451937 0.76 MAOB (0.56) ACHEMAOBMAOANFE2L2RELA
SCHEMBL5793223 0.75 TAAR1 (0.52) TAAR1ACHEIDO1MAOBMAOA
SCHEMBL10783126 0.75 IDO1 (0.55) TAAR1ACHEIDO1MAOBMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129531-B2 Using an isoquinoline compound; alkylation of benzonitrile; reduction ofnitrile to an amine; cyclization BASF AKTIENGESELLSCHAFT (DE) 2012-03-06 US claimed
WO-1997037986-A1 ENDOTHELIN ANTAGONISTS WITH ETHER-LINKED GROUPS WARNER-LAMBERT COMPANY (US) 1997-10-16 WO claimed