Tenocyclidine

Tenocyclidine

SCHEMBL517558

c1csc(C2(N3CCCCC3)CCCCC2)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 10/20 1.00
MEN1 O00255 3/20 1.00
KMT2A Q03164 3/20 1.00
PRCP P42785 2/20 1.00
SLC6A9 P48067 3/20 0.53
SLC6A3 Q01959 2/20 0.53
GRIN1 Q05586 2/20 0.53
GRIN2A Q12879 2/20 0.53
GRIN2B Q13224 2/20 0.53
GRIN2D O15399 1/20 0.53
GRIN3B O60391 1/20 0.53
CYP2B6 P20813 1/20 0.53
SLC6A2 P23975 1/20 0.53
SLC6A4 P31645 1/20 0.53
KCNH2 Q12809 1/20 0.53
GRIN2C Q14957 1/20 0.53
GRIN3A Q8TCU5 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2D6 P10635 1/20 0.53
TSHR P16473 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1742361 1.00 SIGMAR1 (1.00) SIGMAR1MEN1KMT2APRCPSLC6A9
Tenocyclidine SCHEMBL7204633 0.98 SIGMAR1 (0.97) SIGMAR1MEN1KMT2APRCPSLC6A9
Rolicyclidine SCHEMBL15476513 0.91 SIGMAR1 (0.82) SIGMAR1MEN1KMT2APRCPSLC6A9
SCHEMBL7701615 0.88 SIGMAR1 (0.79) SIGMAR1MEN1KMT2APRCPSLC6A9
SCHEMBL7695403 0.87 SIGMAR1 (0.77) SIGMAR1MEN1KMT2APRCPSLC6A9
SCHEMBL29406833 0.85 SIGMAR1 (0.74) SIGMAR1MEN1KMT2APRCPSLC6A9
SCHEMBL7703474 0.84 SIGMAR1 (0.72) SIGMAR1MEN1KMT2APRCPSLC6A9
SCHEMBL8867380 0.84 SIGMAR1 (0.72) SIGMAR1MEN1KMT2APRCPSLC6A9
SCHEMBL8866891 0.84 SIGMAR1 (0.73) SIGMAR1MEN1KMT2APRCPSLC6A9
Tenocyclidine SCHEMBL28321720 0.83 SIGMAR1 (0.68) SIGMAR1MEN1KMT2APRCPSLC6A9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 680 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12539337-B2 Nanostructure conjugates for modulation of location-specific subtypes of receptors and ion channels Molokanova, Elena (US) 2026-02-03 US claimed
EP-4629989-A2 TREATMENT OR PREVENTION OF DEPRESSIVE DISORDERS THROUGH COMBINATION THERAPY Freedom Biosciences, Inc. (US) 2025-10-15 EP claimed
WO-2025111482-A1 COMPLEXING AGENT SALT FORMULATIONS OF PHARMACEUTICAL COMPOUNDS AT LOW STOICHIOMETRIC RATIOS BEXSON BIOMEDICAL, INC. (US) 2025-05-30 WO claimed
US-20250161264-A1 (AMPAR-PAM)-NMDA RECEPTOR ANTAGONIST COMBINATION THERAPY FOR TREATMENT OF MENTAL CONDITIONS AND DISORDERS GILGAMESH PHARMACEUTICALS, INC. 2025-05-22 US claimed
US-20240350433-A1 TREATMENT COMPOSITIONS AND METHODS UNIV YALE (US) 2024-10-24 US claimed
WO-2024123935-A2 TREATMENT OR PREVENTION OF DEPRESSIVE DISORDERS THROUGH COMBINATION THERAPY FREEDOM BIOSCIENCES, INC. (US) 2024-06-13 WO claimed
WO-2024074850-A1 A TREATMENT FOR MENTAL DISORDERS ReWire Therapeutics Limited (GB) 2024-04-11 WO claimed
US-20240066003-A1 NEURODEVELOPMENTAL DISORDER THERAPY ANAVEX LIFE SCIENCES CORP. (US) 2024-02-29 US claimed
WO-2023196234-A1 METHODS, DEVICES, AND SYSTEMS FOR TREATING LENS PROTEIN AGGREGATION DISEASES GLAZIER ALAN NEIL (US) 2023-10-12 WO claimed
US-20230310380-A1 METHODS, DEVICES, AND SYSTEMS FOR TREATING LENS PROTEIN AGGREGATION DISEASES GLAZIER ALAN NEIL (US) 2023-10-05 US claimed
US-20040242848-A1 Mouse/human chimeric anti-phencyclidine antibody and uses thereof NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2004-12-02 US claimed
EP-1438020-A2 TOPICAL COMPOSITIONS AND METHODS FOR TREATING PAIN EpiCept Corporation (US) 2004-07-21 EP claimed
US-20040076648-A1 Topical compositions and methods for treating pain EPICEPT CORPORATION 2004-04-22 US claimed
US-20030082214-A1 Topical compositions and methods for treating pain DISCOVER GROWTH FUND, LLC (VI) 2003-05-01 US claimed
WO-2003015699-A2 TOPICAL COMPOSITIONS AND METHODS FOR TREATING PAIN EPICEPT CORPORATION (US) 2003-02-27 WO claimed
EP-1124553-A1 NEW USE OF GLUTAMATE ANTAGONISTS FOR THE TREATMENT OF CANCER Ikonomidou, Hrissanthi (DE) 2001-08-22 EP claimed
EP-1002535-A1 New use of glutamate antagonists for the treatment of cancer Ikonomidou, Hrissanthi (DE) 2000-05-24 EP claimed
WO-2000024395-A1 NEW USE OF GLUTAMATE ANTAGONISTS FOR THE TREATMENT OF CANCER IKONOMIDOU HRISSANTHI (DE) 2000-05-04 WO claimed
WO-1998010757-A9 THE USE OF FUNCTIONAL N-METHYL-D-ASPARTATE ANTAGONISTS TO AMELIORATE OR PREVENT AMINOGLYCOSIDE-INDUCED OTOTOXICITY 1998-07-23 WO claimed
WO-1998010757-A2 THE USE OF FUNCTIONAL N-METHYL-D-ASPARTATE ANTAGONISTS TO AMELIORATE OR PREVENT AMINOGLYCOSIDE-INDUCED OTOTOXICITY THE GOVERNMENT OF THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1998-03-19 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12539337-B2 Nanostructure conjugates for modulation of location-specific subtypes of receptors and ion channels GRIN2B, GRIN2A, GRIN3A SIGMAR1 123/4885MEN1 3762/4885KMT2A 3507/4885
US-20250161264-A1 (AMPAR-PAM)-NMDA RECEPTOR ANTAGONIST COMBINATION THERAPY FOR TREATMENT OF MENTAL CONDITIONS AND DISORDERS GRIN2A, GRIN1, GRIN3A SIGMAR1 99/4885MEN1 4388/4885KMT2A 611/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.