SCHEMBL5177628

SCHEMBL5177628

COc1ccc(CNS(=O)(=O)c2ccc(-c3nc4cc(OC(N)=O)ccc4[nH]3)cc2)cc1

nearest known ligand 0.72

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 11/20 0.72
TSHR P16473 1/20 0.49
ALDH1A1 P00352 2/20 0.47
CNR1 P21554 3/20 0.47
SLC2A1 P11166 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5177810 0.93 CHEK2 (0.67) CHEK2ALDH1A1
SCHEMBL5178080 0.91 CHEK2 (0.67) CHEK2
SCHEMBL5177601 0.91 CHEK2 (0.66) CHEK2ALDH1A1
SCHEMBL5178049 0.90 CHEK2 (0.67) CHEK2TSHRALDH1A1
SCHEMBL3571821 0.89 CHEK2 (0.86) CHEK2TSHR
SCHEMBL5178184 0.88 CHEK2 (0.68) CHEK2
SCHEMBL5177744 0.87 CHEK2 (0.69) CHEK2ALDH1A1
SCHEMBL5252173 0.86 CHEK2 (0.70) CHEK2
SCHEMBL5176583 0.84 CHEK2 (0.68) CHEK2
SCHEMBL3568934 0.83 CHEK2 (0.70) CHEK2TSHRALDH1A1CNR1SLC2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1613313-B1 2-PHENYL-BENZIMIDAZOL AND 2-PHENYL-IMIDAZO-4,5]-PYRIDINE DERIVATIVES AS CHECKPOINT KINASE CDS1 (CHK2) INHIBITORS FOR THE TREATMENT OF CANCER JANSSEN PHARMACEUTICA NV (BE) 2007-06-06 EP claimed