SCHEMBL5178069

SCHEMBL5178069

Cc1cc(C(=O)NCc2ccc(C(=N)N)cc2[NH])ccc1F

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 13/20 0.51
HTR7 P34969 2/20 0.42
EPHX2 P34913 2/20 0.42
CA2 P00918 1/20 0.41
NR1H4 Q96RI1 1/20 0.41
ROCK2 O75116 1/20 0.40
ROCK1 Q13464 1/20 0.40
PLAU P00749 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5178074 0.89 KLKB1 (0.52) KLKB1EPHX2CA2NR1H4ROCK2
SCHEMBL5178321 0.82 KLKB1 (0.47) KLKB1EPHX2CA2NR1H4ROCK2
SCHEMBL8266479 0.82 F10 (0.48) KLKB1EPHX2ROCK2ROCK1PLAU
SCHEMBL5094014 0.82 CA1 (0.49) KLKB1CA2
Acetic Acid SCHEMBL5178953 0.80 F10 (0.48) KLKB1EPHX2NR1H4PLAU
Hydrochloric Acid SCHEMBL5178223 0.79 F10 (0.53) KLKB1EPHX2ROCK2ROCK1PLAU
SCHEMBL5177725 0.79 KLKB1 (0.44) KLKB1ROCK2ROCK1
SCHEMBL8266177 0.79 F10 (0.52) KLKB1
Hydrochloric Acid SCHEMBL5138361 0.78 F10 (0.52) KLKB1
Hydrochloric Acid SCHEMBL5177719 0.78 KLKB1 (0.44) KLKB1ROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1791810-A1 4-AMINOMETHYL BENZAMIDINE DERIVATIVES AND THEIR USE AS FACTOR VIIA INHIBITORS F. Hoffmann-Roche AG (CH) 2007-06-06 EP disclosed
WO-2006027135-A1 4-AMINOMETHYL BENZAMIDINE DERIVATIVES AND THEIR USE AS FACTOR VIIIA INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2006-03-16 WO disclosed