SCHEMBL5178703

SCHEMBL5178703

CCCN(c1ncc(C(=O)OCC)cn1)c1cc2c(cc1C)C(C)(C)CCC2(C)C

nearest known ligand 0.65

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
RXRA P19793 17/20 0.65
RXRB P28702 15/20 0.65
RXRG P48443 15/20 0.65
PPARG P37231 2/20 0.46
NR1H3 Q13133 1/20 0.46
RARA P10276 4/20 0.41
RARB P10826 4/20 0.41
RARG P13631 3/20 0.41
CYP3A4 P08684 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5179730 0.88 RXRA (0.83) RXRARXRBRXRGPPARGNR1H3
SCHEMBL5179745 0.87 RXRA (0.61) RXRARXRBRXRGPPARGNR1H3
SCHEMBL5180347 0.86 RXRA (0.59) RXRARXRBRXRGPPARGNR1H3
SCHEMBL5179743 0.84 RXRA (0.64) RXRARXRBRXRGPPARGNR1H3
SCHEMBL17049060 0.83 RXRA (0.78) RXRARXRBRXRGPPARGNR1H3
SCHEMBL17049097 0.79 RXRA (1.00) RXRARXRBRXRGPPARGNR1H3
SCHEMBL5179721 0.74 RXRA (0.58) RXRARXRBRXRGPPARGNR1H3
SCHEMBL5180019 0.73 RXRA (0.76) RXRARXRBRXRGPPARGNR1H3
SCHEMBL5180413 0.73 RXRA (0.44) RXRARXRBRXRGPPARGRARA
SCHEMBL5179608 0.73 RXRA (0.76) RXRARXRBRXRGPPARGNR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1180520-B1 PYRIMIDINE CARBOXYLIC ACID DERIVATIVES INST MED MOLECULAR DESIGN INC (JP) 2007-06-20 EP disclosed
US-6869959-B1 Heterocyclic carboxylic acid derivatives INSTITUTE OF MEDICINAL MOLECULAR DESIGN INC. (JP) 2005-03-22 US disclosed
EP-1180520-A1 HETEROCYCLIC CARBOXYLIC ACID DERIVATIVES Institute of Medicinal Molecular Design, Inc. (JP) 2002-02-20 EP disclosed